SCHEMBL16804333

SCHEMBL16804333

CC(C)(O)CN1CCC2(CCN(c3ccnc4c3ccn4Cc3ccc(C(N)=O)cc3)CC2)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.36
MAOB P27338 1/20 0.36
RCOR1 Q9UKL0 1/20 0.36
AKT2 P31751 3/20 0.34
CXCR4 P61073 2/20 0.34
AKT1 P31749 2/20 0.34
NPY2R P49146 1/20 0.32
DRD2 P14416 2/20 0.32
HTR6 P50406 2/20 0.32
GRM2 Q14416 2/20 0.32
METTL3 Q86U44 1/20 0.32
USP7 Q93009 1/20 0.32
GHSR Q92847 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRK1 P41145 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16804413 0.90 HDAC6 (0.41) KDM1AMAOBRCOR1CXCR4
SCHEMBL18125623 0.89 SMN1; SMN2 (0.39) KDM1AMAOBRCOR1CXCR4OPRK1
SCHEMBL16804290 0.87 HDAC6 (0.42)
SCHEMBL16804212 0.87 OPRD1 (0.39) USP7GHSROPRK1CYP3A4CYP2C9
SCHEMBL18125625 0.85 SMN1; SMN2 (0.40) GHSROPRM1OPRK1
SCHEMBL20525344 0.85 DRD2 (0.33) AKT2AKT1DRD2HTR6GRM2
SCHEMBL16804296 0.83 HDAC6 (0.41) KDM1AMAOBRCOR1
SCHEMBL18109007 0.81 MEN1 (0.40) DRD2HTR6
SCHEMBL18108913 0.78 HDAC1 (0.46) KDM1A
SCHEMBL18108961 0.78 CYP11B2 (0.39) OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015087151-A1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2015-06-18 WO disclosed