SCHEMBL20525344

SCHEMBL20525344

CC(C)(O)CN1CC2(CCN(c3ccnc4c3ccn4Cc3ccc(C(N)=O)c(O)c3)CC2)C1

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.33
HTR6 P50406 4/20 0.33
GRM2 Q14416 6/20 0.33
AKT2 P31751 3/20 0.33
AKT1 P31749 2/20 0.33
IRAK4 Q9NWZ3 1/20 0.31
OGA O60502 1/20 0.31
FGFR1 P11362 1/20 0.31
FGFR4 P22455 1/20 0.31
SIRT2 Q8IXJ6 1/20 0.30
SIRT1 Q96EB6 1/20 0.30
SIRT3 Q9NTG7 1/20 0.30
CNR2 P34972 1/20 0.30
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20525329 0.87 GHSR (0.43)
SCHEMBL20525382 0.85 CYP1A2 (0.38) DRD2HTR6
SCHEMBL20525472 0.85 CYP3A4 (0.40) MEN1
SCHEMBL16804333 0.85 KDM1A (0.36) DRD2HTR6GRM2AKT2AKT1
SCHEMBL20525417 0.85 FGFR1 (0.32) FGFR1FGFR4SIRT2SIRT1SIRT3
SCHEMBL20525408 0.83 FAAH (0.38) DRD2HTR6
SCHEMBL20525461 0.82 DGAT1 (0.38) GRM2OGAFGFR1FGFR4CNR2
SCHEMBL20525436 0.82 FGFR1 (0.32) GRM2FGFR1FGFR4
SCHEMBL16804212 0.81 OPRD1 (0.39) MEN1
SCHEMBL16804290 0.81 HDAC6 (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3080125-B1 NOVEL AZAINDOLE DERIVATIVES AS SELECTIVE HISTONE DEACETYLASE (HDAC) INHIBITORS AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME CHONG KUN DANG PHARMACEUTICAL CORP (KR) 2018-10-10 EP disclosed