SCHEMBL1680780

SCHEMBL1680780

O=C(NCc1ccc(Oc2cccc(Br)c2)s1)c1ccc2ncccc2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.48
RAB9A P51151 2/20 0.48
CASP3 P42574 1/20 0.48
SENP8 Q96LD8 1/20 0.48
SENP7 Q9BQF6 1/20 0.48
SENP6 Q9GZR1 1/20 0.48
PLK1 P53350 1/20 0.44
LOX P28300 2/20 0.43
LOXL2 Q9Y4K0 2/20 0.43
ALOX15 P16050 1/20 0.42
HTT P42858 1/20 0.42
HDAC6 Q9UBN7 2/20 0.41
HDAC1 Q13547 2/20 0.41
LMNA P02545 2/20 0.41
EGLN1 Q9GZT9 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.40
TAS1R1 Q7RTX1 1/20 0.40
HDAC2 Q92769 1/20 0.39
HPGD P15428 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1681122 0.90 PLK1 (0.45) NPC1RAB9APLK1LOXLOXL2
SCHEMBL1681352 0.89 MAPK14 (0.49) RAB9APLK1LOXLOXL2ALOX15
SCHEMBL1680976 0.89 EGLN1 (0.47) PLK1LOXLOXL2ALOX15HTT
SCHEMBL1680904 0.89 RAB9A (0.47) NPC1RAB9APLK1LOXLOXL2
SCHEMBL1680909 0.86 LOX (0.44) PLK1LOXLOXL2ALOX15HTT
SCHEMBL1680985 0.86 SPHK2 (0.46) NPC1RAB9APLK1LOXLOXL2
SCHEMBL1680951 0.85 PLK1 (0.46) NPC1RAB9APLK1ALOX15HTT
SCHEMBL1681194 0.85 EGLN1 (0.48) NPC1RAB9APLK1ALOX15HTT
SCHEMBL1680826 0.83 NPC1 (0.47) NPC1RAB9AHTTHDAC1LMNA
SCHEMBL13491542 0.82 ALOX15 (0.54) NPC1RAB9APLK1ALOX15HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110195999-A1 NOVEL ANTIFUNGAL AGENT CONTAINING HETEROCYCLIC COMPOUND NAKAMOTO KAZUTAKA 2011-08-11 US disclosed
US-7932272-B2 Antifungal agent containing heterocyclic compound EISAI R&D MANAGEMENT CO., LTD. (JP) 2011-04-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110195999-A1 NOVEL ANTIFUNGAL AGENT CONTAINING HETEROCYCLIC COMPOUND ERG28, CYP51A1, XPO1 NPC1 170/4885RAB9A 1844/4885CASP3 248/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.