SCHEMBL16824848

SCHEMBL16824848

CN(C)Cc1cc(N)ccc1N1CCOCC1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 7/20 0.58
GAA P10253 5/20 0.58
SMN1; SMN2 Q16637 3/20 0.58
LGMN Q99538 2/20 0.43
ALDH1A1 P00352 3/20 0.42
KDM4E B2RXH2 2/20 0.42
RAD52 P43351 2/20 0.42
LMNA P02545 1/20 0.42
GFER P55789 1/20 0.42
BRAF P15056 1/20 0.42
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
THRB P10828 2/20 0.41
NR4A1 P22736 1/20 0.41
PTK2B Q14289 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
POLB P06746 2/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29949140 1.00 MAPT (0.58) MAPTGAASMN1; SMN2LGMNALDH1A1
SCHEMBL7039460 0.86 MAPT (0.51) MAPTGAASMN1; SMN2ALDH1A1KDM4E
SCHEMBL24630249 0.84 MAPT (0.61) MAPTGAASMN1; SMN2LGMNALDH1A1
SCHEMBL29769230 0.84 MAPT (0.61) MAPTGAASMN1; SMN2LGMNALDH1A1
SCHEMBL17536983 0.84 SMN1; SMN2 (0.50) MAPTGAASMN1; SMN2ALDH1A1KDM4E
SCHEMBL16454989 0.82 MAPT (0.58) MAPTGAASMN1; SMN2LGMNALDH1A1
SCHEMBL29889006 0.82 CCR5 (0.47) MAPTGAASMN1; SMN2ALDH1A1LMNA
SCHEMBL27159794 0.82 CCR5 (0.47) MAPTGAASMN1; SMN2ALDH1A1LMNA
SCHEMBL13455200 0.81 MAPT (0.61) MAPTGAASMN1; SMN2LGMNALDH1A1
SCHEMBL188672 0.81 MAPT (0.61) MAPTGAASMN1; SMN2LGMNALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12466841-B2 Substituted pyrrolo[3,4-c]pyridines as HPK1 antagonists Nimbus Saturn, Inc. (US) 2025-11-11 US disclosed
US-12071442-B2 Substituted pyrrolo[3,4-c]pyridines as HPK1 antagonists Nimbus Saturn, Inc. (US) 2024-08-27 US disclosed
US-20240190895-A1 SUBSTITUTED PYRROLO[3,4-c]PYRIDINES AS HPK1 ANTAGONISTS CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED (GB) 2024-06-13 US disclosed
CN-117377673-A HPK1 antagonists and uses thereof 林伯士萨顿公司 2024-01-09 CN disclosed
US-20220363695-A1 HPK1 ANTAGONISTS AND USES THEREOF Nimbus Saturn, Inc. 2022-11-17 US disclosed
US-9850247-B2 Pyrimidopyrimidinones useful as Wee-1 kinase inhibitors ALMAC HOUSE (GB) 2017-12-26 US disclosed
EP-3083625-B1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS ALMAC DISCOVERY LTD (GB) 2017-11-01 EP disclosed
US-20160318936-A1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2016-11-03 US disclosed
EP-3083625-A1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS Almac Discovery Limited (GB) 2016-10-26 EP disclosed
WO-2015092431-A1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2015-06-25 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220363695-A1 HPK1 ANTAGONISTS AND USES THEREOF PDXK, HIPK1, PCK1 MAPT 3895/4885GAA 905/4885SMN1; SMN2 3277/4885
US-20160318936-A1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS WEE1, WEE2, NME1 MAPT 3728/4885GAA 1730/4885SMN1; SMN2 4422/4885
US-12466841-B2 Substituted pyrrolo[3,4-c]pyridines as HPK1 antagonists PDXK, HIPK1, HIPK3 MAPT 3393/4885GAA 2502/4885SMN1; SMN2 3266/4885
US-12071442-B2 Substituted pyrrolo[3,4-c]pyridines as HPK1 antagonists PDXK, HIPK1, PGK1 MAPT 3822/4885GAA 2572/4885SMN1; SMN2 3520/4885
US-20240190895-A1 SUBSTITUTED PYRROLO[3,4-c]PYRIDINES AS HPK1 ANTAGONISTS PDXK, HIPK1, HIPK3 MAPT 3393/4885GAA 2502/4885SMN1; SMN2 3266/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.