SCHEMBL1683803

SCHEMBL1683803

COc1cc(C=O)c(-c2csc(-c3ncccn3)n2)c(OC)c1OC

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 19/20 0.51
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1683842 0.85 CYP19A1 (0.48) CYP19A1KDM4E
SCHEMBL1683981 0.80 MAPT (0.41) CYP19A1KDM4EALDH1A1
SCHEMBL2544743 0.78 MAPT (0.40) CYP19A1
SCHEMBL2543254 0.78 TUBB4A (0.42) KDM4EALDH1A1
Hydrochloric Acid SCHEMBL2547764 0.77 MAPT (0.39) CYP19A1
Hydrochloric Acid SCHEMBL2539879 0.76 HDAC3 (0.39) CYP19A1KDM4E
SCHEMBL2743529 0.72 ALDH1A1 (0.57) KDM4EALDH1A1TSHRTDP1
SCHEMBL15225838 0.71 ALDH1A1 (0.50) KDM4EALDH1A1
SCHEMBL4038581 0.70 ALDH1A1 (0.47) KDM4EALDH1A1
SCHEMBL1683776 0.68 EGFR (0.58) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2303021-A2 COMPOUNDS FOR THE TREATMENT OF CANCER University of Tennessee Research Foundation (US) 2011-04-06 EP disclosed
WO-2010074776-A2 COMPOUNDS FOR THE TREATMENT OF CANCER THE UNIVERSITY OF TENNESSEE RESEARCH FOUNDATION (US) 2010-07-01 WO disclosed