SCHEMBL16840720

SCHEMBL16840720

CNc1cc(C(F)(F)F)nc(C)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.50
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
NOS3 P29474 1/20 0.41
NOS2 P35228 1/20 0.41
HPGD P15428 3/20 0.41
ATM Q13315 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
ALDH1A1 P00352 3/20 0.38
KMT2A Q03164 3/20 0.38
MAPT P10636 2/20 0.38
MEN1 O00255 2/20 0.38
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
CRHBP P24387 1/20 0.37
CYP2C19 P33261 1/20 0.37
CRHR2 Q13324 1/20 0.37
RAB9A P51151 2/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31453693 0.82 ALDH1A1 (0.45) KDM4EHSP90AA1HSP90AB1HPGDATM
SCHEMBL25846980 0.82 NOS3 (0.42) KDM4ENOS3NOS2ALDH1A1KMT2A
SCHEMBL10271825 0.80 HSP90AA1 (0.52) KDM4EHSP90AA1HSP90AB1HPGDATM
SCHEMBL22247617 0.78 KDM4E (0.49) KDM4EHSP90AA1HSP90AB1NOS3NOS2
SCHEMBL17812892 0.78 NOS3 (0.54) NOS3NOS2ALDH1A1MAPTCYP3A4
SCHEMBL25065895 0.76 KDM4E (0.46) KDM4EHSP90AA1HSP90AB1NOS3NOS2
SCHEMBL14927263 0.74 HSP90AA1 (0.63) KDM4EHSP90AA1HSP90AB1HPGDATM
Hydrochloric Acid SCHEMBL28210241 0.73 KDM4E (0.44) KDM4EHSP90AA1HSP90AB1HPGDATM
SCHEMBL27776507 0.73 SDHB (0.54) KDM4EHPGDALDH1A1KMT2AMAPT
Ammonia Solution, Strong SCHEMBL15795498 0.72 HSP90AA1 (0.61) KDM4EHSP90AA1HSP90AB1HPGDATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015091584-A1 THIAZOLOPYRIDINE COMPOUNDS, COMPOSITIONS AND THEIR USE AS TYK2 KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2015-06-25 WO disclosed