SCHEMBL16848725

SCHEMBL16848725

CCCN(C)c1ccc(C=O)nc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 2/20 0.39
TRPV1 Q8NER1 3/20 0.37
KCNH2 Q12809 2/20 0.36
ALDH1A1 P00352 3/20 0.34
ALDH3A1 P30838 3/20 0.34
ALDH1A3 P47895 3/20 0.34
MAPT P10636 2/20 0.34
KCNJ1 P48048 1/20 0.33
CYP2A6 P11509 1/20 0.32
CYP2A13 Q16696 1/20 0.32
KDM4E B2RXH2 3/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
THRB P10828 1/20 0.32
MAPK1 P28482 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
ATM Q13315 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
AOC3 Q16853 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8196798 0.78 KCNH2 (0.54) KCNH2ALDH1A1MAPTKCNJ1CYP2A6
SCHEMBL24991834 0.77 ALDH1A1 (0.55) KCNH2ALDH1A1ALDH3A1ALDH1A3MAPT
SCHEMBL7865566 0.74 MAPT (0.40) HCAR3TRPV1ALDH1A1MAPTMEN1
SCHEMBL12781461 0.74 HCAR3 (0.38) HCAR3TRPV1MAPT
SCHEMBL12201383 0.73 ALDH1A1 (0.59) ALDH1A1ALDH3A1ALDH1A3MAPTCYP2A6
SCHEMBL2767198 0.71 KCNH2 (0.37) KCNH2ALDH1A1KCNJ1CYP2A6CYP2A13
SCHEMBL6741043 0.71 MAPT (0.49) HCAR3TRPV1ALDH1A1MAPTMEN1
SCHEMBL15198856 0.71 KCNJ1 (0.39) KCNH2ALDH1A1KCNJ1CYP2A6CYP2A13
SCHEMBL231541 0.70 LTC4S (0.39) KCNH2
SCHEMBL7089251 0.68 SMN1; SMN2 (0.44) ALDH1A1MAPTKCNJ1KDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2886534-A1 Benzene or thiophene derivative and use thereof as VAP-1 inhibitor R-Tech Ueno, Ltd. (JP) 2015-06-24 EP disclosed