SCHEMBL1688010

SCHEMBL1688010

CCCCOc1c(N(Cc2ccccc2)Cc2ccccc2)cc(N(C)C)c(C)c1C(=O)Oc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ATM Q13315 1/20 0.41
NR3C1 P04150 8/20 0.40
TSPO P30536 1/20 0.39
CYP2D6 P10635 2/20 0.38
MMP9 P14780 1/20 0.37
MMP13 P45452 1/20 0.37
ADAM17 P78536 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
NPC1 O15118 1/20 0.37
LMNA P02545 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
HSD17B10 Q99714 1/20 0.37
PGR P06401 1/20 0.37
NR3C2 P08235 1/20 0.37
AR P10275 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6128436 0.88 NR3C1 (0.39) MEN1KMT2AATMNR3C1TSPO
SCHEMBL1687998 0.76 FAAH (0.41) KMT2ACYP2D6NPC1LMNATSHR
SCHEMBL113438 0.76 TSPO (0.41) KMT2ANR3C1TSPOLMNA
SCHEMBL13417394 0.75 FAAH (0.42) KMT2ACYP2D6NPC1LMNATSHR
SCHEMBL13417245 0.74 KMT2A (0.35) MEN1KMT2AATMLMNATSHR
SCHEMBL17849881 0.74 FAAH (0.34) MEN1KMT2ANR3C1MMP9MMP13
SCHEMBL17849906 0.73 FAAH (0.33) MEN1KMT2ANR3C1CYP2D6MMP9
SCHEMBL9288716 0.73 FAAH (0.42) KMT2ACYP2D6NPC1LMNATSHR
SCHEMBL10107486 0.72 LMNA (0.41) KMT2ACYP2D6NPC1LMNATSHR
SCHEMBL9286322 0.72 FAAH (0.38) KMT2ACYP2D6NPC1LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047907-A9 SYNTHESIS OF C5-SUBSTITUTED TETRACYCLINES, USES THEREOF, AND INTERMEDIATES THERETO PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-09-27 WO disclosed
WO-2012047907-A1 SYNTHESIS OF C5-SUBSTITUTED TETRACYCLINES, USES THEREOF, AND INTERMEDIATES THERETO PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-04-12 WO disclosed