SCHEMBL16888149

SCHEMBL16888149

CCS(=O)(=O)c1ccc(CC(=O)Nc2nc3c(s2)CN(c2ccccc2)CC3)cc1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RORC P51449 14/20 0.55
PIK3CG P48736 1/20 0.53
RORB Q92753 1/20 0.52
SLC27A1 Q6PCB7 1/20 0.51
ALDH1A1 P00352 2/20 0.50
LMNA P02545 2/20 0.50
GAA P10253 2/20 0.49
ESR1 P03372 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2D6 P10635 1/20 0.49
MAPT P10636 1/20 0.49
CYP2C9 P11712 1/20 0.49
HPGD P15428 1/20 0.49
CYP2C19 P33261 1/20 0.49
KMT2A Q03164 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16888128 0.90 RORC (0.50) RORCPIK3CGRORBALDH1A1LMNA
SCHEMBL16888126 0.89 RORC (0.53) RORCRORBALDH1A1GAAESR1
SCHEMBL16888130 0.88 RORC (0.50) RORCRORBALDH1A1LMNAGAA
SCHEMBL16879789 0.81 LMNA (0.73) RORCRORBALDH1A1LMNAGAA
SCHEMBL12307656 0.80 PIK3CG (0.78) PIK3CGSLC27A1ALDH1A1LMNAGAA
SCHEMBL16888127 0.79 PIK3CG (0.45) RORCPIK3CGSLC27A1ALDH1A1GAA
SCHEMBL16888045 0.79 RORC (0.44) RORCPIK3CGRORBALDH1A1GAA
SCHEMBL19772202 0.79 RORC (0.56) RORCRORB
SCHEMBL19772097 0.79 RORC (0.56) RORCRORB
SCHEMBL16888129 0.78 ALDH1A1 (0.44) RORCPIK3CGRORBALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015101928-A1 FUSED THIOPHENE AND THIAZOLE DERIVATIVES AS ROR GAMMA MODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2015-07-09 WO disclosed