SCHEMBL1688906

SCHEMBL1688906

O=c1c2cn(-c3ccccc3)nc2nc(-c2ccc(N3CCOCC3)cc2Cl)n1-c1ccc(Cl)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.45
IDO2 Q6ZQW0 1/20 0.45
MAT2A P31153 1/20 0.43
CNR1 P21554 3/20 0.41
ALDH1A1 P00352 3/20 0.41
MEN1 O00255 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
KMT2A Q03164 2/20 0.41
HSD17B10 Q99714 2/20 0.41
CNR2 P34972 1/20 0.41
USP2 O75604 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
HIF1A Q16665 1/20 0.41
GAA P10253 4/20 0.40
TSHR P16473 2/20 0.40
KDM4E B2RXH2 2/20 0.40
MAPK1 P28482 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1688884 0.89 CNR1 (0.45) TDO2IDO2MAT2ACNR1ALDH1A1
SCHEMBL1688973 0.87 KDM4E (0.46) TDO2IDO2CNR1ALDH1A1MEN1
SCHEMBL5611633 0.83 MAPT (0.43) CNR1ALDH1A1MEN1CYP1A2CYP2C9
SCHEMBL1688941 0.83 PTGS2 (0.41) ALDH1A1MEN1CYP1A2CYP2C9CYP2C19
SCHEMBL1688982 0.81 KDM4E (0.43) CNR1CNR2KDM4EMAPK1PTGS2
SCHEMBL5611689 0.81 KDM4E (0.43) TDO2IDO2MAT2ACNR1ALDH1A1
SCHEMBL5611929 0.81 ALDH1A1 (0.43) TDO2IDO2MAT2AALDH1A1MEN1
SCHEMBL1753603 0.80 MAPT (0.58) ALDH1A1KMT2ATSHRKDM4EMAPK1
SCHEMBL1688942 0.78 CNR1 (0.43) MAT2ACNR1KMT2ACNR2KDM4E
SCHEMBL5611629 0.77 SMN1; SMN2 (0.41) CNR1ALDH1A1MEN1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807429-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM, LLC (BM) 2007-07-18 EP claimed
WO-2006047516-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2006-05-04 WO claimed