SCHEMBL1689259

SCHEMBL1689259

N#Cc1cccc(C(C(N)=O)(C(N)=O)c2cccc(C#N)c2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.44
GSK3B P49841 2/20 0.44
ENPP2 Q13822 1/20 0.42
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
KMT2A Q03164 1/20 0.41
GRIN2D O15399 2/20 0.41
GRIN3B O60391 2/20 0.41
GRIN1 Q05586 2/20 0.41
GRIN2A Q12879 2/20 0.41
GRIN2B Q13224 2/20 0.41
GRIN2C Q14957 2/20 0.41
GRIN3A Q8TCU5 2/20 0.41
PTPN5 P54829 1/20 0.40
XDH P47989 1/20 0.40
SLC22A12 Q96S37 1/20 0.40
KCNN4 O15554 1/20 0.40
NOTUM Q6P988 1/20 0.39
PDK1 Q15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6165966 0.81 KCNN4 (0.59) KIF11MAPTKMT2AGRIN2DGRIN3B
SCHEMBL6163962 0.78 KCNN4 (0.55) KIF11MEN1ALDH1A1MAPTKMT2A
SCHEMBL7101543 0.78 KCNN4 (0.55) KIF11MEN1ALDH1A1MAPTKMT2A
SCHEMBL3937789 0.74 SGK1 (0.47) KIF11GSK3BENPP2MEN1ALDH1A1
SCHEMBL22285654 0.74 PTPN5 (0.46) KIF11GSK3BENPP2MEN1ALDH1A1
SCHEMBL29675909 0.73 VNN1 (0.46) GSK3BMEN1ALDH1A1MAPTKMT2A
Trifluoroacetic Acid SCHEMBL27502598 0.72 FFAR1 (0.52) MEN1MAPTKMT2APTPN5PDK1
Bicarbonate SCHEMBL11598627 0.72 GSK3B (0.55) GSK3BENPP2MEN1ALDH1A1MAPT
SCHEMBL4593887 0.72 PARP1 (0.52) KIF11MAPTKMT2APTPN5KCNN4
SCHEMBL16892944 0.72 PARP1 (0.52) KIF11MEN1ALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896395-B1 MODIFIED MALONATE DERIVATIVES MERCK SHARP & DOHME (US) 2015-07-15 EP disclosed