SCHEMBL1690386

SCHEMBL1690386

CC(C)(C)C(=Cc1cnc2c(c1)CC(C)(C)C(=O)N2)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
RAMP1 O60894 4/20 0.33
CALCRL Q16602 4/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16403839 1.00 RAMP1 (0.33) RAMP1CALCRL
SCHEMBL1690385 1.00 RAMP1 (0.33) RAMP1CALCRL
SCHEMBL1092657 0.81
SCHEMBL1092659 0.81
SCHEMBL3611131 0.79 RAB9A (0.40)
SCHEMBL3611126 0.79 RAB9A (0.40)
SCHEMBL1093388 0.79
SCHEMBL1093390 0.79
SCHEMBL1255043 0.77
SCHEMBL1255042 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3004099-A1 TETRAHYDROPYRIDINE DERIVATIVES AS FabI INHIBITORS Aurigene Discovery Technologies Limited (IN) 2016-04-13 EP disclosed
WO-2014195844-A1 TETRAHYDROPYRIDINE DERIVATIVES AS FabI INHIBITORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2014-12-11 WO disclosed
US-20140107106-A1 THERAPEUTIC AGENTS, AND METHODS OF MAKING AND USING THE SAME AFFINIUM PHARMACEUTICALS, INC. (CA) 2014-04-17 US disclosed
US-8450307-B2 Therapeutic agents, and methods of making and using the same AFFINIUM PHARMACEUTICALS, INC. (CA) 2013-05-28 US disclosed
US-20120010127-A1 Compositions Comprising Multiple Bioactive Agents, and Methods of Using the Same BERMAN JUDD M (CA) 2012-01-12 US disclosed
US-20100093705-A1 Therapeutic agents, and methods of making and using the same DEBIOPHARM INTERNATIONAL SA (CH) 2010-04-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100093705-A1 Therapeutic agents, and methods of making and using the same MCL1, DHFR, ANXA5 RAMP1 4827/4885CALCRL 1886/4885
US-20120010127-A1 Compositions Comprising Multiple Bioactive Agents, and Methods of Using the Same DBI, SERPINB1, CTSF RAMP1 4540/4885CALCRL 3743/4885
US-20140107106-A1 THERAPEUTIC AGENTS, AND METHODS OF MAKING AND USING THE SAME MCL1, DHFR, ANXA5 RAMP1 4827/4885CALCRL 1886/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.