SCHEMBL1695015

SCHEMBL1695015

Nc1c(F)cccc1C=O

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 4/20 0.57
MEN1 O00255 1/20 0.46
LMNA P02545 1/20 0.46
THRB P10828 1/20 0.46
BLM P54132 1/20 0.46
KMT2A Q03164 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
NFE2L2 Q16236 3/20 0.41
ALDH1A1 P00352 2/20 0.38
TSHR P16473 1/20 0.38
TRIM24 O15164 1/20 0.38
TRIM33 Q9UPN9 1/20 0.38
CYP2A6 P11509 1/20 0.35
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TLR2 O60603 1/20 0.34
TLR1 Q15399 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30106737 1.00 ERN1 (0.57) ERN1MEN1LMNATHRBBLM
SCHEMBL29139204 0.83 KMT2A (0.58) ERN1MEN1LMNATHRBBLM
SCHEMBL13887136 0.77 NFE2L2 (0.41) ERN1NFE2L2ALDH1A1GRIN2DGRIN3B
SCHEMBL17023603 0.77 ALDH1A1 (0.44) ERN1MEN1LMNATHRBBLM
SCHEMBL154794 0.76 ERN1 (0.61) ERN1MEN1LMNATHRBBLM
SCHEMBL1655785 0.76 TDP1 (0.50) ERN1MEN1LMNATHRBBLM
SCHEMBL30039913 0.75
SCHEMBL29540911 0.75
SCHEMBL20465749 0.75
SCHEMBL87096 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 41 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118894867-A Preparation of 12-fluorocamptothecin derivative and application thereof in anti-tumor aspect 兰州大学 2024-11-05 CN claimed
CN-107522766-A One kind has ursolic acid quinolyl hydrazide derivatives of antitumor activity and its preparation method and application 南京林业大学 2017-12-29 CN claimed
EP-4622967-A1 COMPOUNDS THAT INHIBIT PKMYT1 Exelixis, Inc. (US) 2025-10-01 EP disclosed
US-20250171431-A1 HETEROCYCLIC INHIBITORS OF IGF-1R FOR TREATMENT OF DISEASE HORIZON THERAPEUTICS IRELAND DAC (IE) 2025-05-29 US disclosed
CN-119585247-A Bicyclic heterocyclic amide inhibitors of nav1.8 for the treatment of pain 赛特温治疗公司 2025-03-07 CN disclosed
EP-4514789-A1 <SUP2/>? <SUB2/>?V?BICYCLIC HETEROCYCLIC AMIDE INHIBITORS OF NA1.8 FOR THE TREATMENT OF PAIN SiteOne Therapeutics, Inc. (US) 2025-03-05 EP disclosed
US-12220421-B2 Inhibitors of C. difficile spore germination THE BOARDS OF REGENTS OF THE NEVADA SYSTEM OF HIGHER EDUCATION ON BEHALF OF THE UNIVERSITY OF NEVADA, LAS (US) 2025-02-11 US disclosed
WO-2025030163-A1 HETEROCYCLIC INHIBITORS OF IGF-1R FOR TREATMENT OF DISEASE HORIZON THERAPEUTICS IRELAND DAC (IE) 2025-02-06 WO disclosed
CN-118894867-A Preparation of 12-fluorocamptothecin derivative and application thereof in anti-tumor aspect 兰州大学 2024-11-05 CN disclosed
EP-4398890-A2 INHIBITORS OF C. DIFFICILE SPORE GERMINATION Abel-Santos, Ernesto (US) 2024-07-17 EP disclosed
WO-2024112853-A1 COMPOUNDS THAT INHIBIT PKMYT1 EXELIXIS, INC. (US) 2024-05-30 WO disclosed
US-20100331306-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2010-12-30 US disclosed
US-20100331306-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2010-12-30 US disclosed
WO-2010151740-A2 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2010-12-29 WO disclosed
WO-2010151740-A2 HETEROCYCLIC COMPOUNDS AND THEIR USES AMGEN INC. (US) 2010-12-29 WO disclosed
US-5532374-A Method of preparation of bis-quinolines HITACHI CHEMICAL COMPANY, LTD. (JP) 1996-07-02 US disclosed
EP-0093611-B2 Composite plasmid AJINOMOTO KK (JP) 1995-03-22 EP disclosed
EP-0093611-B1 COMPOSITE PLASMID AJINOMOTO CO., INC. (JP) 1987-07-22 EP disclosed
US-4514502-A DRUG RESISTANCE AJINOMOTO CO., INC. (JP) 1985-04-30 US disclosed
EP-0093611-A1 Composite plasmid AJINOMOTO CO., INC. (JP) 1983-11-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12220421-B2 Inhibitors of C. difficile spore germination CDC37, SI, DAD1 ERN1 2577/4885MEN1 4513/4885LMNA 4332/4885
US-20100331306-A1 HETEROCYCLIC COMPOUNDS AND THEIR USES MCL1, BCL9, MALT1 ERN1 3475/4885MEN1 1596/4885LMNA 2321/4885
US-20250171431-A1 HETEROCYCLIC INHIBITORS OF IGF-1R FOR TREATMENT OF DISEASE IGF1R, TRHR, TSHR ERN1 2399/4885MEN1 160/4885LMNA 3056/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.