SCHEMBL1697008

SCHEMBL1697008

O=C(O)c1cccc2ccc(O)nc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
LMNA P02545 1/20 0.50
ALOX12 P18054 1/20 0.50
KDM4E B2RXH2 4/20 0.49
KMT2A Q03164 2/20 0.49
NR4A1 P22736 1/20 0.47
NR4A2 P43354 1/20 0.47
NR4A3 Q92570 1/20 0.47
PARP1 P09874 4/20 0.46
HSD17B10 Q99714 2/20 0.46
LDHA P00338 1/20 0.43
ALOX15 P16050 1/20 0.43
MEN1 O00255 1/20 0.42
TSHR P16473 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
HPGD P15428 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
HMGB1 P09429 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30170409 0.81 KDM4E (0.68) ALDH1A1LMNAKDM4EKMT2ANR4A1
SCHEMBL7143621 0.81 KDM4E (0.68) ALDH1A1LMNAKDM4EKMT2ANR4A1
SCHEMBL29412561 0.79 PARP1 (0.72) ALDH1A1ALOX12KDM4EKMT2ANR4A1
SCHEMBL27908511 0.79 ALDH1A1 (0.49) ALDH1A1LMNAALOX12KDM4EKMT2A
SCHEMBL1032809 0.79 SLC40A1 (0.49) ALDH1A1LMNAALOX12KDM4EKMT2A
SCHEMBL5319765 0.79 PARP1 (0.72) ALDH1A1ALOX12KDM4EKMT2ANR4A1
SCHEMBL28798022 0.79 KDM4E (0.66) ALDH1A1LMNAKDM4EKMT2AALOX15
SCHEMBL27283354 0.79 KDM4E (0.66) ALDH1A1LMNAKDM4EKMT2AALOX15
SCHEMBL5149194 0.78 PARP1 (0.70) ALDH1A1ALOX12KDM4EKMT2ANR4A1
SCHEMBL21816896 0.78 PARP1 (0.70) ALDH1A1ALOX12KDM4EKMT2ANR4A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2273992-B1 QUINOLINES AND RELATED ANALOGS AS SIRTUIN MODULATORS GLAXOSMITHKLINE LLC (US) 2016-05-25 EP disclosed
WO-2012003145-A2 THERAPEUTIC AGENTS FOR OCULAR HYPERTENSION ALLERGAN, INC. (US) 2012-01-05 WO disclosed