SCHEMBL27908511

SCHEMBL27908511

O=C(O)c1cccc2ccc(Br)nc12

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
NR4A1 P22736 1/20 0.46
NR4A2 P43354 1/20 0.46
NR4A3 Q92570 1/20 0.46
PARP1 P09874 5/20 0.45
LMNA P02545 1/20 0.45
ALOX12 P18054 1/20 0.45
HSD17B10 Q99714 1/20 0.44
KDM4E B2RXH2 2/20 0.43
KMT2A Q03164 1/20 0.43
ALOX15 P16050 1/20 0.41
CDC25B P30305 1/20 0.41
KEAP1 Q14145 1/20 0.41
HPGD P15428 1/20 0.41
DHODH Q02127 1/20 0.40
PTPN1 P18031 1/20 0.40
WDR5 P61964 1/20 0.39
MMP2 P08253 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27891655 0.84 PARP1 (0.44) ALDH1A1PARP1LMNAALOX12KDM4E
SCHEMBL29103150 0.84 PARP1 (0.47) ALDH1A1PARP1KDM4EKMT2A
SCHEMBL30170409 0.79 KDM4E (0.68) ALDH1A1NR4A1NR4A2NR4A3LMNA
SCHEMBL7143621 0.79 KDM4E (0.68) ALDH1A1NR4A1NR4A2NR4A3LMNA
SCHEMBL1697008 0.79 ALDH1A1 (0.50) ALDH1A1NR4A1NR4A2NR4A3PARP1
SCHEMBL5319765 0.78 PARP1 (0.72) ALDH1A1NR4A1NR4A2NR4A3PARP1
SCHEMBL1032809 0.78 SLC40A1 (0.49) ALDH1A1NR4A1NR4A2NR4A3PARP1
SCHEMBL28798022 0.78 KDM4E (0.66) ALDH1A1LMNAKDM4EKMT2AALOX15
SCHEMBL27283354 0.78 KDM4E (0.66) ALDH1A1LMNAKDM4EKMT2AALOX15
SCHEMBL29412561 0.78 PARP1 (0.72) ALDH1A1NR4A1NR4A2NR4A3PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102942524-B Preparation method of quinoline derivative BEIJING VAGEAN TECHNOLOGY CO LTD 2014-12-31 CN disclosed
CN-102942524-A Preparation method of quinoline derivative BEIJING VAGEAN SCIENCE & TECHNOLOGY CO LTD 2013-02-27 CN disclosed