SCHEMBL1698216

SCHEMBL1698216

c1cnc2c(c1)CCCC2C1CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
CXCR4 P61073 11/20 0.39
CYP2D6 P10635 3/20 0.39
SIGMAR1 Q99720 2/20 0.38
CYP3A4 P08684 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1698200 0.91 KDM4E (0.39) HDAC1HDAC6CXCR4CYP2D6KDM4E
SCHEMBL29587352 0.84 HTR2A (0.36) CYP2D6CYP3A4KDM4EGAA
SCHEMBL9672362 0.76 CXCR4 (0.46) CXCR4CYP2D6
SCHEMBL2083952 0.75 CXCR4 (0.43) HDAC1HDAC6CXCR4CYP2D6CYP3A4
SCHEMBL10612034 0.75 HDAC1 (0.41) HDAC1HDAC6CXCR4CYP2D6CYP3A4
SCHEMBL23850650 0.75 HDAC1 (0.41) HDAC1HDAC6CXCR4CYP2D6
SCHEMBL13857919 0.75 HDAC1 (0.41) HDAC1HDAC6CXCR4CYP2D6
SCHEMBL12891529 0.75 CYP2D6 (0.43) HDAC1HDAC6CXCR4CYP2D6
SCHEMBL5021376 0.75 P2RX7 (0.45) HDAC1HDAC6CXCR4CYP2D6
SCHEMBL24804097 0.75 HDAC1 (0.41) HDAC1HDAC6CXCR4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8933231-B2 Organic compounds GIVAUDAN SA 2015-01-13 US disclosed
US-8933231-B2 Organic compounds GIVAUDAN SA 2015-01-13 US disclosed
US-8933231-B2 Organic compounds GIVAUDAN SA 2015-01-13 US disclosed
CN-102946741-B Organic compounds GIVAUDAN SA 2014-05-14 CN disclosed
US-20130129655-A1 Organic Compounds GIVAUDAN SA (CH) 2013-05-23 US disclosed
US-20130129655-A1 Organic Compounds GIVAUDAN SA (CH) 2013-05-23 US disclosed
US-20130129655-A1 Organic Compounds GIVAUDAN SA (CH) 2013-05-23 US disclosed
EP-2584916-A1 ORGANIC COMPOUNDS Givaudan SA (CH) 2013-05-01 EP disclosed
WO-2011161163-A1 ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2011-12-29 WO disclosed
WO-2011161163-A1 ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2011-12-29 WO disclosed
WO-2011160254-A1 ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2011-12-29 WO disclosed
WO-2011160254-A1 ORGANIC COMPOUNDS GIVAUDAN SA (CH) 2011-12-29 WO disclosed
EP-1465889-A4 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS WITH ENHANCED EFFICACY ANORMED INC (CA) 2008-05-14 EP disclosed
EP-1465889-A1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS WITH ENHANCED EFFICACY AnorMED Inc. (CA) 2004-10-13 EP disclosed
WO-2003055876-A1 CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS WITH ENHANCED EFFICACY ANORMED INC. (CA) 2003-07-10 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130129655-A1 Organic Compounds C9, C5, TRPA1 HDAC1 939/4885HDAC6 1775/4885CXCR4 1601/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.