SCHEMBL16986933

SCHEMBL16986933

O=C(O)c1n[nH]cc1Nc1ccccc1[N+](=O)[O-]

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.55
ASPH Q12797 1/20 0.55
KDM8 Q8N371 1/20 0.55
ALDH1A1 P00352 5/20 0.51
MAPK1 P28482 3/20 0.51
TDP1 Q9NUW8 3/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
CASP7 P55210 1/20 0.51
AKR1C3 P42330 4/20 0.49
AKR1C2 P52895 4/20 0.49
MAPT P10636 7/20 0.47
MEN1 O00255 6/20 0.47
KMT2A Q03164 6/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
RAB9A P51151 3/20 0.47
GAA P10253 5/20 0.47
PKM P14618 1/20 0.47
AKR1B1 P15121 2/20 0.45
AKR1C4 P17516 2/20 0.45
AKR1C1 Q04828 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2801162 0.81 CYP1A2 (0.53) ALDH1A1MEN1KMT2ASMN1; SMN2RAB9A
SCHEMBL10917448 0.76 FABP4 (0.46) KDM4EALDH1A1MAPK1TDP1AKR1C3
SCHEMBL11279444 0.76 MAPT (0.54) KDM4EASPHKDM8ALDH1A1MAPK1
SCHEMBL182687 0.76 LMNA (0.41) KDM4EASPHKDM8TDP1L3MBTL1
SCHEMBL397773 0.75 MAPK1 (0.77) ALDH1A1MAPK1TDP1L3MBTL1CASP7
SCHEMBL453183 0.75 AKR1C3 (0.68) KDM4EASPHKDM8ALDH1A1MAPK1
SCHEMBL5181747 0.71 MAPK1 (0.57) KDM4EASPHKDM8ALDH1A1MAPK1
SCHEMBL2875877 0.71 KDM4E (1.00) KDM4EASPHKDM8ALDH1A1MAPK1
SCHEMBL2877327 0.71 KDM4E (1.00) KDM4EASPHKDM8ALDH1A1MAPK1
SCHEMBL953645 0.70 MAPT (0.58) KDM4EALDH1A1MAPK1TDP1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1845973-B1 PHARMACEUTICAL COMPOUNDS ASTEX THERAPEUTICS LTD (GB) 2015-08-12 EP disclosed