SCHEMBL1699084

SCHEMBL1699084

CCc1c(C)cnc2c1[nH]c(=O)n2-c1ccc(Oc2nc3cccnc3n2C)cc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 5/20 0.39
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
POLB P06746 1/20 0.37
PABPC1 P11940 1/20 0.37
PDE10A Q9Y233 5/20 0.36
TP53 P04637 1/20 0.35
LMNA P02545 2/20 0.34
DCTPP1 Q9H773 1/20 0.34
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
PDE4B Q07343 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699248 0.90 DRD1 (0.38) DRD1MEN1KMT2APOLBPABPC1
SCHEMBL1699098 0.89 DRD1 (0.44) DRD1MEN1KMT2APOLBPABPC1
SCHEMBL1699092 0.88 DRD1 (0.38) DRD1MEN1KMT2APOLBPABPC1
SCHEMBL1699557 0.86 HDAC1 (0.37) DRD1MEN1KMT2APOLBPABPC1
SCHEMBL1699111 0.86 PDE10A (0.36) DRD1MEN1KMT2APOLBPABPC1
SCHEMBL14889112 0.82 DRD1 (0.38) DRD1MEN1KMT2APOLBPABPC1
SCHEMBL1699476 0.80 PDE10A (0.36) DRD1PDE10ALMNAHDAC1HDAC6
SCHEMBL1699250 0.77 PDE10A (0.36) DRD1MEN1KMT2APDE10ALMNA
SCHEMBL1699226 0.75 ALDH1A1 (0.35) MEN1KMT2APDE10ALMNA
SCHEMBL14333706 0.74 ALDH1A1 (0.37) DRD1KMT2APOLBLMNAHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed