SCHEMBL1699358

SCHEMBL1699358

CCCCOC(C(=O)O)c1c(C)cc2ccccc2c1Cl

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.38
KCNH2 Q12809 2/20 0.37
MCL1 Q07820 3/20 0.37
PPARG P37231 2/20 0.36
PPARA Q07869 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
PLA2G2A P14555 1/20 0.36
DHODH Q02127 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27903964 0.85 GPR84 (0.39) KCNH2PPARGPPARAMEN1KMT2A
SCHEMBL27903971 0.78 GRM2 (0.34) PPARGPPARAMEN1KMT2APLA2G2A
SCHEMBL1699348 0.78 PSIP1 (0.39) CYP3A4LMNASMN1; SMN2
SCHEMBL1699271 0.78 PSIP1 (0.39) CYP3A4LMNASMN1; SMN2
SCHEMBL27903966 0.78 CXCR5 (0.33) PPARGPPARAMEN1KMT2APLA2G2A
SCHEMBL27921784 0.76 ESR1 (0.41) KCNH2PPARGPPARACNR2ESR1
SCHEMBL27921912 0.76 GPR84 (0.41) KCNH2PPARGPPARAMEN1KMT2A
SCHEMBL27903976 0.76 DHODH (0.37) PPARGPPARADHODHCNR1
SCHEMBL1699401 0.74 PTPN1 (0.36) ALOX5KCNH2PPARGPPARAMEN1
SCHEMBL27921762 0.74 CTRC (0.39) PPARGPPARADHODHCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2588450-A1 NAPHT- 2 -YLACETIC ACID DERIVATIVES TO TREAT AIDS Gilead Sciences, Inc. (US) 2013-05-08 EP disclosed
WO-2012003497-A1 NAPHT- 2 -YLACETIC ACID DERIVATIVES TO TREAT AIDS GILEAD SCIENCES, INC. (US) 2012-01-05 WO disclosed