SCHEMBL17004202

SCHEMBL17004202

c1cc2cc(-c3nnc(OC4C5CC6CC4CN(C6)C5)s3)ccc2s1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 6/20 0.38
KCNH2 Q12809 4/20 0.38
CHRNB2 P17787 2/20 0.38
CHRNB4 P30926 2/20 0.38
CHRNA3 P32297 2/20 0.38
CHRNA4 P43681 2/20 0.38
DYRK1A Q13627 1/20 0.34
KDM1A O60341 1/20 0.34
CA12 O43570 3/20 0.31
ENPP1 P22413 1/20 0.31
CA2 P00918 2/20 0.31
SIGMAR1 Q99720 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17004358 0.80 CHRNA7 (0.56) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL3833132 0.80 MGAM (0.39) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL17004237 0.80 CHRNB2 (0.39) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
Abt-126 SCHEMBL16033886 0.80 CHRNB2 (0.49) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
Abt-126 SCHEMBL878680 0.80 CHRNB2 (0.49) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
Abt-126 SCHEMBL16782423 0.80 CHRNB2 (0.49) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
Abt-126 SCHEMBL12695541 0.80 CHRNB2 (0.49) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL17004229 0.79 CHRNA7 (0.48) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL17004231 0.79 CHRNA7 (0.49) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3
SCHEMBL17004239 0.78 CHRNA7 (0.47) CHRNA7KCNH2CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099795-B1 AZAADAMANTANE DERIVATIVES AND THEIR USES AS NICOTINIC ACETYLCHOLINE RECEPTORS LIGANDS ABBVIE BAHAMAS LTD (BS) 2015-08-19 EP disclosed