SCHEMBL17004231

SCHEMBL17004231

c1cc2ccc(-c3nnc(OC4C5CC6CC4CN(C6)C5)s3)cc2[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 8/20 0.49
CHRNB2 P17787 3/20 0.49
CHRNA4 P43681 3/20 0.49
CHRNB4 P30926 2/20 0.49
CHRNA3 P32297 2/20 0.49
GUSB P08236 6/20 0.37
KCNH2 Q12809 4/20 0.35
S1PR1 P21453 1/20 0.33
MPO P05164 1/20 0.32
LCK P06239 1/20 0.31
BTK Q06187 1/20 0.31
HTR3A P46098 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC7 Q8WUI4 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17004358 0.93 CHRNA7 (0.56) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17004208 0.82 CHRNA7 (0.37) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17004237 0.80 CHRNB2 (0.39) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL3833132 0.80 MGAM (0.39) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
Abt-126 SCHEMBL16782423 0.80 CHRNB2 (0.49) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
Abt-126 SCHEMBL16033886 0.80 CHRNB2 (0.49) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
Abt-126 SCHEMBL878680 0.80 CHRNB2 (0.49) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
Abt-126 SCHEMBL12695541 0.80 CHRNB2 (0.49) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17004202 0.79 CHRNA7 (0.38) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17004209 0.78 CHRNA7 (0.38) CHRNA7CHRNB2CHRNA4CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099795-B1 AZAADAMANTANE DERIVATIVES AND THEIR USES AS NICOTINIC ACETYLCHOLINE RECEPTORS LIGANDS ABBVIE BAHAMAS LTD (BS) 2015-08-19 EP disclosed