SCHEMBL17004209

SCHEMBL17004209

c1cc(-c2nnc(OC3C4CC5CC3CN(C5)C4)s2)c2cc[nH]c2c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 6/20 0.38
CHRNB2 P17787 2/20 0.37
CHRNB4 P30926 2/20 0.37
CHRNA3 P32297 2/20 0.37
CHRNA4 P43681 2/20 0.37
KCNH2 Q12809 2/20 0.36
PIK3CD O00329 3/20 0.33
MTOR P42345 1/20 0.33
S1PR1 P21453 1/20 0.32
LRRK2 Q5S007 1/20 0.31
IDH2 P48735 1/20 0.30
ATR Q13535 1/20 0.30
PIK3CA P42336 1/20 0.30
PIK3CB P42338 1/20 0.30
PIK3CG P48736 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30
HTR1A P08908 1/20 0.30
ROCK2 O75116 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17004236 0.83 CHRNA7 (0.38) CHRNA7KCNH2PIK3CDMTORLRRK2
SCHEMBL17004231 0.78 CHRNA7 (0.49) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL17004358 0.78 CHRNA7 (0.56) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
Abt-126 SCHEMBL16782423 0.77 CHRNB2 (0.49) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
Abt-126 SCHEMBL12695541 0.77 CHRNB2 (0.49) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
Abt-126 SCHEMBL878680 0.77 CHRNB2 (0.49) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL1110502 0.76 CHRNA7 (0.44) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL17004223 0.72 KDM4E (0.43) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL3833132 0.72 MGAM (0.39) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL17004237 0.72 CHRNB2 (0.39) CHRNA7CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099795-B1 AZAADAMANTANE DERIVATIVES AND THEIR USES AS NICOTINIC ACETYLCHOLINE RECEPTORS LIGANDS ABBVIE BAHAMAS LTD (BS) 2015-08-19 EP disclosed