SCHEMBL17004249

SCHEMBL17004249

Clc1ccncc1OC1C2CC3CC1CN(C3)C2

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.34
CHRNB4 P30926 2/20 0.34
CHRNA3 P32297 2/20 0.34
CHRNA7 P36544 2/20 0.34
CHRNA4 P43681 2/20 0.34
ADRA2A P08913 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA2C P18825 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR2B P41595 1/20 0.32
CYP17A1 P05093 1/20 0.32
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17004259 0.83 CHRNB2 (0.38) CHRNB2CHRNB4CHRNA3CHRNA4CHRM2
SCHEMBL17004295 0.75 CHRNB2 (0.41) CHRNB2CHRNA4ADRA2AADRA2BADRA2C
SCHEMBL3825645 0.74 CHRNB2 (0.41) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL17004242 0.72 CHRM2 (0.54) CHRM2CHRM1
SCHEMBL17004213 0.71 CHRNB2 (0.41) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL17004311 0.71 TRPC3 (0.35) CHRM2CHRM1
SCHEMBL17004218 0.70 CHRNB2 (0.42) CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL17004329 0.69 LNPEP (0.35) ADRA2AADRA2BADRA2CHTR2AHTR2C
SCHEMBL17004243 0.69 S1PR4 (0.33) CHRNB4CHRNA3CHRNA7
SCHEMBL17004220 0.69 CHRNB2 (0.36) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099795-B1 AZAADAMANTANE DERIVATIVES AND THEIR USES AS NICOTINIC ACETYLCHOLINE RECEPTORS LIGANDS ABBVIE BAHAMAS LTD (BS) 2015-08-19 EP disclosed