SCHEMBL17004259

SCHEMBL17004259

Cc1ccncc1OC1C2CC3CC1CN(C3)C2

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.38
CHRNA4 P43681 2/20 0.38
GPR119 Q8TDV5 1/20 0.33
SOST Q9BQB4 1/20 0.32
SIRT3 Q9NTG7 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
CHRM2 P08172 1/20 0.30
CHRM1 P11229 1/20 0.30
SSTR4 P31391 1/20 0.30
CHRNB4 P30926 1/20 0.30
CHRNA3 P32297 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17004249 0.83 CHRNB2 (0.34) CHRNB2CHRNA4CHRM2CHRM1CHRNB4
SCHEMBL17004242 0.72 CHRM2 (0.54) CHRM2CHRM1
SCHEMBL17004311 0.71 TRPC3 (0.35) CHRM2CHRM1
SCHEMBL17004233 0.70 NAAA (0.32) CHRM2CHRM1
SCHEMBL17004295 0.69 CHRNB2 (0.41) CHRNB2CHRNA4GPR119CHRM1
SCHEMBL17004243 0.69 S1PR4 (0.33) CHRNB4CHRNA3
SCHEMBL17004288 0.69 FLT3 (0.34) CHRNB2CHRNA4CHRNB4CHRNA3
SCHEMBL17004220 0.69 CHRNB2 (0.36) CHRNB2CHRNA4CHRM2CHRM1CHRNB4
SCHEMBL23021681 0.69 CHRNB2 (0.47) CHRNB2CHRNA4GPR119SIRT3TDP1
SCHEMBL17004285 0.69 HSD11B1 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2099795-B1 AZAADAMANTANE DERIVATIVES AND THEIR USES AS NICOTINIC ACETYLCHOLINE RECEPTORS LIGANDS ABBVIE BAHAMAS LTD (BS) 2015-08-19 EP disclosed