SCHEMBL1702794

SCHEMBL1702794

Cc1ccc(F)c(NC(=O)Nc2ccc(-c3cncc4[nH]nc(N)c34)cc2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 19/20 1.00
FLT3 P36888 11/20 1.00
CSF1R P07333 9/20 1.00
FLT4 P35916 9/20 1.00
KIT P10721 9/20 1.00
LYN P07948 8/20 1.00
FLT1 P17948 8/20 1.00
BLK P51451 7/20 1.00
LCK P06239 7/20 1.00
SRC P12931 6/20 1.00
FYN P06241 5/20 1.00
AURKA O14965 5/20 0.78
AURKB Q96GD4 5/20 0.78
ROCK2 O75116 4/20 0.78
MET P08581 4/20 0.78
RPS6KB1 P23443 4/20 0.78
CSNK1D P48730 4/20 0.78
ROCK1 Q13464 4/20 0.78
ABL1 P00519 3/20 0.78
PDGFRB P09619 3/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13523218 0.90 KDR (0.82) KDRFLT3CSF1RFLT4KIT
Linifanib SCHEMBL93804 0.88 KDR (1.00) KDRFLT3CSF1RFLT4KIT
Linifanib SCHEMBL29375368 0.88 KDR (1.00) KDRFLT3CSF1RFLT4KIT
SCHEMBL1703142 0.87 KDR (1.00) KDRFLT3CSF1RFLT4KIT
SCHEMBL1702799 0.87 KDR (1.00) KDRFLT3CSF1RFLT4KIT
SCHEMBL12426039 0.87 KDR (0.77) KDRFLT3CSF1RFLT4KIT
Linifanib SCHEMBL1880038 0.87 KDR (0.98) KDRFLT3CSF1RFLT4KIT
Linifanib SCHEMBL2239943 0.85 KDR (0.94) KDRFLT3CSF1RFLT4KIT
SCHEMBL233874 0.84 KDR (1.00) KDRFLT3CSF1RFLT4KIT
SCHEMBL1703302 0.83 KDR (0.79) KDRFLT3CSF1RFLT4KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807424-B1 NOVEL KINASE INHIBITORS ABBOTT LAB (US) 2012-04-18 EP claimed
EP-1807424-A2 NOVEL KINASE INHIBITORS ABBOTT LABORATORIES (US) 2007-07-18 EP claimed
US-20060178378-A1 Novel kinase inhibitors ABBVIE INC. 2006-08-10 US claimed
WO-2006050109-A2 NOVEL KINASE INHIBITORS ABBOTT LABORATORIES (US) 2006-05-11 WO claimed
EP-1807424-B1 NOVEL KINASE INHIBITORS ABBOTT LAB (US) 2012-04-18 EP disclosed
US-7812166-B2 Kinase inhibitors ABBOTT LABORATORIES (US) 2010-10-12 US disclosed
US-20100004306-A1 PIGF-1 Assay and kits and components thereof ABBOTT LABORATORIES (US) 2010-01-07 US disclosed
US-20060178378-A1 Novel kinase inhibitors ABBVIE INC. 2006-08-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060178378-A1 Novel kinase inhibitors ABL1, MAP3K19, MAP3K20 KDR 434/4885FLT3 79/4885CSF1R 1265/4885
US-20100004306-A1 PIGF-1 Assay and kits and components thereof PGF, FLT1, HDGF KDR 9/4885FLT3 773/4885CSF1R 126/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.