SCHEMBL1703637

SCHEMBL1703637

Nc1cnn(Cc2cccc(Cl)c2)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.63
MEN1 O00255 2/20 0.63
MAPT P10636 3/20 0.56
LMNA P02545 2/20 0.56
KLKB1 P03952 2/20 0.53
L3MBTL1 Q9Y468 3/20 0.51
TDP1 Q9NUW8 2/20 0.51
POLB P06746 1/20 0.51
ALDH1A1 P00352 1/20 0.48
PKM P14618 1/20 0.48
ITK Q08881 1/20 0.46
SIGMAR1 Q99720 1/20 0.45
PNMT P11086 1/20 0.44
KDM4E B2RXH2 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44
SCD5 Q86SK9 1/20 0.44
ALK Q9UM73 1/20 0.44
TSHR P16473 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29442842 1.00 KMT2A (0.63) KMT2AMEN1MAPTLMNAKLKB1
SCHEMBL14712472 0.85 MEN1 (0.68) KMT2AMEN1MAPTLMNAKLKB1
SCHEMBL950986 0.83 MAPT (0.67) KMT2AMEN1MAPTLMNAKLKB1
SCHEMBL712713 0.82 MAPT (0.70) KMT2AMEN1MAPTLMNAKLKB1
Hydrochloric Acid SCHEMBL17822246 0.82 MAPT (0.70) KMT2AMEN1MAPTLMNAKLKB1
SCHEMBL1703331 0.81 MEN1 (0.68) KMT2AMEN1MAPTLMNAKLKB1
SCHEMBL19087042 0.81 L3MBTL1 (0.51) KMT2AMEN1MAPTLMNAKLKB1
SCHEMBL16096120 0.81 L3MBTL1 (0.55) KMT2AMEN1MAPTLMNAKLKB1
SCHEMBL14699255 0.81 KMT2A (0.63) KMT2AMEN1MAPTLMNAL3MBTL1
SCHEMBL3616273 0.81 MAPT (0.65) KMT2AMEN1MAPTLMNAKLKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 22 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12180221-B2 Compounds and uses thereof JANSSEN PHARMACEUTICA NV (BE) 2024-12-31 US disclosed
CN-118084801-A Compounds and uses thereof 詹森药业有限公司 2024-05-28 CN disclosed
CN-118084800-A Compounds and uses thereof 詹森药业有限公司 2024-05-28 CN disclosed
CN-112312913-B Compounds and uses thereof 詹森药业有限公司 2024-03-08 CN disclosed
US-20230078764-A1 COMPOUNDS AND USES THEREOF JANSSEN PHARMACEUTICA NV (BE) 2023-03-16 US disclosed
US-20220298168-A1 COMPOUNDS AND USES THEREOF JANSSEN PHARMACEUTICA NV (BE) 2022-09-22 US disclosed
CN-114174273-A Compounds and uses thereof 优曼尼蒂治疗公司 2022-03-11 CN disclosed
CN-112566636-A Compound and use thereof 优曼尼蒂治疗公司 2021-03-26 CN disclosed
EP-3784234-A1 COMPOUNDS AND USES THEREOF Yumanity Therapeutics, Inc. (US) 2021-03-03 EP disclosed
US-10919885-B2 Compounds and uses thereof YUMANITY THERAPEUTICS, INC. (US) 2021-02-16 US disclosed
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
US-20190330198-A1 COMPOUNDS AND USES THEREOF JANSSEN PHARMACEUTICA NV (BE) 2019-10-31 US disclosed
US-20190330198-A1 COMPOUNDS AND USES THEREOF JANSSEN PHARMACEUTICA NV (BE) 2019-10-31 US disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed
US-8426408-B2 Pyrimidine inhibitors of kinases ABBVIE INC. (US) 2013-04-23 US disclosed
CN-102498110-A 2- (LH-pyrazol-4-ylamino) -pyrimidine as kinase inhibitors ABBOTT LAB 2012-06-13 CN disclosed
EP-2440548-A1 2- ( LH-PYRAZOL-4 -YLAMINO ) -PYRIMIDINE AS KINASE INHIBITORS Abbott Laboratories (US) 2012-04-18 EP disclosed
US-20100317680-A1 PYRIMIDINE INHIBITORS OF KINASES ABBOTT LABORATORIES (US) 2010-12-16 US disclosed
WO-2010144468-A1 2- ( LH-PYRAZOL-4 -YLAMINO ) -PYRIMIDINE AS KINASE INHIBITORS ABBOTT LABORATORIES (US) 2010-12-16 WO disclosed
US-20100041696-A1 Compounds SMITHKLINE BEECHAM CORPORATION 2010-02-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100317680-A1 PYRIMIDINE INHIBITORS OF KINASES AURKA, AURKC, AURKB KMT2A 849/4885MEN1 1727/4885MAPT 2310/4885
US-20100041696-A1 Compounds CYP11B2, SCD, CYP3A5 KMT2A 3500/4885MEN1 3499/4885MAPT 3377/4885
US-20230078764-A1 COMPOUNDS AND USES THEREOF NLN, BDNF, NQO1 KMT2A 587/4885MEN1 191/4885MAPT 101/4885
US-10919885-B2 Compounds and uses thereof NLN, ACHE, CLN6 KMT2A 2479/4885MEN1 1807/4885MAPT 22/4885
US-20220298168-A1 COMPOUNDS AND USES THEREOF NLN, ACHE, CLN6 KMT2A 2479/4885MEN1 1807/4885MAPT 22/4885
US-12180221-B2 Compounds and uses thereof NLN, ACHE, CLN6 KMT2A 2479/4885MEN1 1807/4885MAPT 22/4885
US-20190330198-A1 COMPOUNDS AND USES THEREOF NLN, ACHE, CLN6 KMT2A 2479/4885MEN1 1807/4885MAPT 22/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.