SCHEMBL1703908

SCHEMBL1703908

COC(=O)Cc1ccc(CN2CCN(C(=O)O)[C@](C)(Cc3ccccc3)C2)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.43
CYP2D6 P10635 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
LMNA P02545 2/20 0.42
SIGMAR1 Q99720 2/20 0.42
KDM4E B2RXH2 2/20 0.41
HDAC4 P56524 1/20 0.40
KCNH2 Q12809 1/20 0.40
HDAC1 Q13547 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
TSHR P16473 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
POLB P06746 1/20 0.39
NR3C1 P04150 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1703971 0.84 ALDH1A1 (0.51) ALDH1A1CYP2D6SMN1; SMN2LMNASIGMAR1
SCHEMBL1704763 0.80 CYP4F2 (0.38) ALDH1A1CYP2D6SMN1; SMN2LMNASIGMAR1
SCHEMBL1633895 0.78 KDM4E (0.51) ALDH1A1CYP2D6SMN1; SMN2LMNASIGMAR1
SCHEMBL2007650 0.76 POLB (0.39) ALDH1A1CYP2D6LMNAKDM4ETSHR
SCHEMBL14813579 0.74 GAA (0.50) ALDH1A1CYP2D6SMN1; SMN2LMNASIGMAR1
SCHEMBL1188920 0.74 MEN1 (0.48) ALDH1A1SMN1; SMN2KDM4EHTTMEN1
SCHEMBL7364364 0.74 DRD4 (0.59) SMN1; SMN2LMNAKDM4EHDAC4HDAC1
SCHEMBL1704155 0.74 MLNR (0.60) ALDH1A1CYP2D6KCNH2KMT2APOLB
SCHEMBL1704529 0.74 MLNR (0.60) ALDH1A1CYP2D6KCNH2KMT2APOLB
SCHEMBL25244127 0.73 SMN1; SMN2 (0.53) ALDH1A1CYP2D6SMN1; SMN2LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed