SCHEMBL1704763

SCHEMBL1704763

COC(=O)Cc1ccc(CN2CCN(C(=O)O)[C@@](C)(C(C)(C)C)C2)cc1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.37
ALDH1A1 P00352 4/20 0.37
CYP2D6 P10635 2/20 0.37
SIGMAR1 Q99720 1/20 0.36
LMNA P02545 3/20 0.36
MAPT P10636 2/20 0.36
LIPE Q05469 1/20 0.36
FAAH O00519 1/20 0.35
KDM4E B2RXH2 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704591 0.88 CHRM2 (0.37) ALDH1A1CYP2D6SIGMAR1KDM4E
SCHEMBL377425 0.84 RAB9A (0.40) SMN1; SMN2ALDH1A1LMNAMAPTFAAH
SCHEMBL377693 0.84 RAB9A (0.40) SMN1; SMN2ALDH1A1LMNAMAPTFAAH
SCHEMBL377823 0.83 LMNA (0.44) SMN1; SMN2ALDH1A1SIGMAR1LMNAKDM4E
SCHEMBL377467 0.83 LMNA (0.44) SMN1; SMN2ALDH1A1SIGMAR1LMNAKDM4E
SCHEMBL3565835 0.82 RAB9A (0.41) SMN1; SMN2ALDH1A1SIGMAR1LMNAMAPT
SCHEMBL377528 0.81 KDM4E (0.53) SMN1; SMN2ALDH1A1LMNAMAPTKDM4E
SCHEMBL377869 0.81 KDM4E (0.53) SMN1; SMN2ALDH1A1LMNAMAPTKDM4E
SCHEMBL1703908 0.80 ALDH1A1 (0.43) SMN1; SMN2ALDH1A1CYP2D6SIGMAR1LMNA
SCHEMBL1632683 0.75 KDM4E (0.48) SMN1; SMN2ALDH1A1SIGMAR1FAAHKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed