SCHEMBL1633895

SCHEMBL1633895

C[C@]1(Cc2ccccc2)CN(Cc2cccc(Br)c2)CCN1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
FAAH O00519 1/20 0.50
POLB P06746 2/20 0.48
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
TDP1 Q9NUW8 1/20 0.45
SIGMAR1 Q99720 1/20 0.44
ALDH1A1 P00352 4/20 0.43
HTT P42858 1/20 0.43
LMNA P02545 1/20 0.42
MAPK1 P28482 2/20 0.42
NPSR1 Q6W5P4 1/20 0.42
DRD4 P21917 2/20 0.40
NTRK1 P04629 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C19 P33261 1/20 0.39
MBTD1 Q05BQ5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1703971 0.88 ALDH1A1 (0.51) KDM4EFAAHPOLBKMT2AMEN1
SCHEMBL1632683 0.82 KDM4E (0.48) KDM4EFAAHPOLBKMT2AMEN1
SCHEMBL1703908 0.78 ALDH1A1 (0.43) KDM4EPOLBKMT2AMEN1SMN1; SMN2
SCHEMBL1631552 0.77 CHRM3 (0.40) DRD4
SCHEMBL2007650 0.76 POLB (0.39) KDM4EPOLBKMT2AMEN1ALDH1A1
SCHEMBL5619307 0.75 OPRM1 (0.40) SMN1; SMN2ALDH1A1CYP2D6
SCHEMBL1188920 0.74 MEN1 (0.48) KDM4EKMT2AMEN1SMN1; SMN2TDP1
SCHEMBL3047497 0.73 KDM4E (0.71) KDM4EFAAHPOLBKMT2AMEN1
SCHEMBL14813579 0.73 GAA (0.50) KDM4EPOLBKMT2AMEN1SMN1; SMN2
SCHEMBL1704166 0.70 KDM4E (0.40) KDM4EPOLBKMT2AMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7932247-B2 M3 muscarinic acetylcholine receptor antagonists GLAXO GROUP LIMITED (GB) 2011-04-26 US disclosed