SCHEMBL17049367

SCHEMBL17049367

Brc1ccc(OCc2ccccc2)c(-c2cc(Br)ccc2OCc2ccccc2)c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 5/20 0.56
SLC6A4 P31645 1/20 0.56
MAOB P27338 1/20 0.56
ALDH1A1 P00352 3/20 0.55
USP28 Q96RU2 1/20 0.55
USP25 Q9UHP3 1/20 0.55
RAB9A P51151 1/20 0.55
HTT P42858 2/20 0.54
PTGER1 P34995 4/20 0.53
PTGDR2 Q9Y5Y4 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
CYP2C9 P11712 1/20 0.51
LMNA P02545 1/20 0.50
PTPN1 P18031 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11297633 0.91 PTGDR2 (0.63) CCR5SLC6A4MAOBALDH1A1USP28
SCHEMBL368071 0.87 SLC6A4 (0.66) CCR5SLC6A4MAOBALDH1A1USP28
SCHEMBL31644088 0.87 SLC6A4 (0.66) CCR5SLC6A4MAOBALDH1A1USP28
SCHEMBL7898169 0.85 RAB9A (0.59) CCR5SLC6A4MAOBALDH1A1USP28
SCHEMBL30835101 0.85 RAB9A (0.59) CCR5SLC6A4MAOBALDH1A1USP28
SCHEMBL5690733 0.85 PTGER1 (0.53) CCR5SLC6A4MAOBALDH1A1USP28
SCHEMBL28286296 0.85 CCR5 (0.55) CCR5SLC6A4MAOBALDH1A1USP28
SCHEMBL30835001 0.85 CCR5 (0.55) CCR5SLC6A4MAOBALDH1A1USP28
SCHEMBL3724105 0.82 MEN1 (0.59) CCR5SLC6A4MAOBALDH1A1USP28
SCHEMBL3713861 0.82 CCR5 (0.54) CCR5SLC6A4MAOBALDH1A1USP28

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015127941-A1 QUALITATIVE STRUCTURE ACTIVITY RELATIONSHIP (QSAR) OF NEW ORGANIC COMPOUNDS SYNTHESIZED BY STILLE CROSS COUPLING REACTION WITH ANTITUMOR ACTIVITY ABOU ELSAOUD YASMINE MOHAMED HASHEM EZZ EL DIN (EG) 2015-09-03 WO disclosed