SCHEMBL1705264

SCHEMBL1705264

COc1cc2c(cc1OC)CNC2

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.59
MAPT P10636 1/20 0.59
ALDH1A1 P00352 3/20 0.46
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
MAOA P21397 5/20 0.42
TSHR P16473 1/20 0.42
KDM4E B2RXH2 3/20 0.42
CHRNA7 P36544 2/20 0.42
MAOB P27338 2/20 0.42
SLC6A4 P31645 1/20 0.42
RAB9A P51151 1/20 0.41
GLA P06280 1/20 0.39
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30040451 1.00 CYP3A4 (0.59) CYP3A4MAPTALDH1A1HTR2AHTR2C
Hydrochloric Acid SCHEMBL31193341 0.97 CYP3A4 (0.56) CYP3A4MAPTALDH1A1HTR2AHTR2C
Hydrochloric Acid SCHEMBL9871800 0.97 CYP3A4 (0.56) CYP3A4MAPTALDH1A1HTR2AHTR2C
SCHEMBL6122379 0.84 POLB (0.47) CYP3A4MAPTALDH1A1HTR2AHTR2C
SCHEMBL29788066 0.84 HTR2A (0.61) CYP3A4MAPTHTR2AHTR2CHTR2B
SCHEMBL382917 0.84 HTR2C (0.50) CYP3A4MAPTHTR2AHTR2CHTR2B
SCHEMBL8794833 0.84 CHRNA7 (0.49) CYP3A4MAPTALDH1A1MAOACHRNA7
SCHEMBL329913 0.84 HTR2A (0.61) CYP3A4MAPTHTR2AHTR2CHTR2B
SCHEMBL30677786 0.84 HTR2C (0.67) CYP3A4MAPTALDH1A1HTR2AHTR2C
SCHEMBL13028005 0.84 MAPT (0.43) CYP3A4MAPTALDH1A1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 53 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0186187-A2 Cephalosporin derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1986-07-02 EP claimed
WO-2024149360-A1 BIQUATERNARY AMMONIUM SALT COMPOUND AND PHARMACEUTICAL APPLICATION THEREOF 西藏海思科制药有限公司 2024-07-18 WO disclosed
CN-116987021-A Novel isoindoline derivative with anti-tumor effect as well as preparation method and application thereof 北京中医药大学 2023-11-03 CN disclosed
EP-4212528-A1 BENZO OXYGEN-CONTAINING HETEROCYCLIC COMPOUND AND MEDICAL APPLICATION THEREOF AB Pharma Ltd. (CN) 2023-07-19 EP disclosed
US-20230183197-A1 INHIBITORS OF MLH1 AND/OR PMS2 FOR CANCER TREATMENT Neophore Limited (GB) 2023-06-15 US disclosed
CN-115286616-A Tetrahydroisoquinoline and isoindoline compound capable of binding sigma-2 receptor, preparation method and application thereof 北京师范大学 2022-11-04 CN disclosed
CN-107849047-B Biphenyl derivative, preparation method and medical application thereof 四川海思科制药有限公司 2021-01-15 CN disclosed
EP-3153515-B1 COMPOUNDS FOR INHIBITING HEPATITIS C VIRUS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF AB PHARMA LTD (CN) 2020-08-12 EP disclosed
WO-2020108688-A1 PYRROLOPYRIDINE DERIVATIVES AND THEIR USE FOR NUCLEAR-MEDICAL IMAGING HELMHOLTZ-ZENTRUM DRESDEN-ROSSENDORF E.V. (DE) 2020-06-04 WO disclosed
WO-2020029980-A1 SMAD3 INHIBITORS MOEXA PHARMACEUTICALS LIMITED (CN) 2020-02-13 WO disclosed
US-5561141-A POTENTIATE ACTIVITY OF ANTITUMOR AGENTS AMERICAN CYANAMID COMPANY (US) 1996-10-01 US disclosed
US-5550149-A SULFUR-CONTAINING COMPOUNDS THAT ARE EFFECTIVE IN POTENTIATING THE ACTIVITY OF CHEMOTHERAPEUTIC ANTI-CANCER AGENTS BY INCREASING SENSITIVITY OF MULTI-DRUG RESISTANT CELLS AMERICAN CYANAMID COMPANY (US) 1996-08-27 US disclosed
US-5387685-A MDR reversal agents AMERICAN CYANAMID COMPANY 1995-02-07 US disclosed
EP-0634401-A1 MDR reversal agents AMERICAN CYANAMID COMPANY (US) 1995-01-18 EP disclosed
US-4987235-A Isoindoline derivatives and processes for their preparation BANYU PHARMACEUTICAL CO., LTD. (JP) 1991-01-22 US disclosed
US-4958029-A Process for the production of isoindoline derivatives, novel intermediates and process for their production BANYU PHARMACEUTICAL CO., LTD. (JP) 1990-09-18 US disclosed
EP-0275064-A2 Process for the production of isoindoline derivatives, novel intermediates and process for their production Banyu Pharmaceutical Co., Ltd. (JP) 1988-07-20 EP disclosed
EP-0227986-A1 Isoindoline derivatives and processes for their preparation BANYU PHARMACEUTICAL CO., LTD. (JP) 1987-07-08 EP disclosed
US-4677100-A ANTIBIOTICS BANYU PHARMACEUTICAL CO., LTD. (JP) 1987-06-30 US disclosed
EP-0186187-A2 Cephalosporin derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1986-07-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230183197-A1 INHIBITORS OF MLH1 AND/OR PMS2 FOR CANCER TREATMENT MSH2, PMS2, MSH6 CYP3A4 3288/4885MAPT 3491/4885ALDH1A1 1817/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.