SCHEMBL17067451

SCHEMBL17067451

CC(C)(C)OC(=O)c1sccc1CCN=NN

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
CA14 Q9ULX7 1/20 0.33
ALDH1A1 P00352 2/20 0.32
KMT2A Q03164 3/20 0.31
MAPT P10636 3/20 0.31
NPC1 O15118 1/20 0.31
KDM4E B2RXH2 2/20 0.30
CYP1A2 P05177 2/20 0.30
POLB P06746 1/20 0.30
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
NR3C2 P08235 1/20 0.30
MEN1 O00255 2/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13141391 0.82 KMT2A (0.35) LMNACA12CA1CA2CA9
SCHEMBL4730278 0.79 KMT2A (0.36) LMNACA12CA1CA2CA9
SCHEMBL11389305 0.76 FABP4 (0.37) LMNACA12CA1CA2CA9
SCHEMBL632529 0.76 KMT2A (0.36) LMNAALDH1A1KMT2ANPC1KDM4E
SCHEMBL13141386 0.72 CTSS (0.36) LMNAALDH1A1KMT2AMAPTNPC1
SCHEMBL11389102 0.70 MAPT (0.46) LMNAALDH1A1KMT2AMAPTNPC1
SCHEMBL28220747 0.69 KMT2A (0.36) ALDH1A1KMT2ANPC1KDM4ECYP1A2
SCHEMBL632902 0.69 PKM (0.49) ALDH1A1MAPTNPC1POLBGAA
SCHEMBL5725289 0.67 POLB (0.46) LMNACA12CA1CA2CA9
SCHEMBL23142285 0.67 TDP1 (0.43) CA12CA1CA2CA9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2149561-B1 TETRAHYDROISOQUINOLIN-1-ONE DERIVATIVE OR SALT THEREOF SELDAR PHARMA INC (US) 2015-09-09 EP disclosed