SCHEMBL170730

SCHEMBL170730

Cc1cccc(Oc2ccnc(C(=O)N(C)C)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 2/20 0.50
HSD17B2 P37059 2/20 0.50
RAF1 P04049 4/20 0.47
BRAF P15056 1/20 0.46
MGLL Q99685 1/20 0.46
ALDH1A1 P00352 2/20 0.45
LYN P07948 1/20 0.44
LMNA P02545 1/20 0.43
GRM5 P41594 1/20 0.42
GCK P35557 1/20 0.42
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6014158 0.86 RAF1 (0.54) HSD17B1HSD17B2RAF1BRAFMGLL
SCHEMBL9926359 0.84 LMNA (0.50) HSD17B1HSD17B2ALDH1A1LYNLMNA
SCHEMBL257972 0.83 MAPT (0.48) RAF1BRAFALDH1A1LYNLMNA
SCHEMBL24310884 0.82 KDR (0.48) ALDH1A1LYNGRM5GCKMAPT
SCHEMBL170881 0.81 ALDH1A1 (0.45) HSD17B1HSD17B2ALDH1A1LYNLMNA
SCHEMBL167783 0.81 KDR (0.58) RAF1BRAFALDH1A1LYN
SCHEMBL9926365 0.80 ALDH1A1 (0.44) HSD17B1HSD17B2ALDH1A1LYNLMNA
SCHEMBL620695 0.79 RAF1 (0.53) RAF1BRAFALDH1A1MAPTSMN1; SMN2
SCHEMBL4947098 0.78 ALDH1A1 (0.44) RAF1ALDH1A1MAPTSMN1; SMN2
SCHEMBL18780870 0.76 RAF1 (0.48) HSD17B1HSD17B2RAF1BRAFALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426122-A1 Methylene urea derivative as RAF kinasse inhibitors Merck Patent GmbH (DE) 2012-03-07 EP disclosed
EP-1158985-B1 OMEGA-CARBOXY ARYL SUBSTITUTED DIPHENYL UREAS AS p38 KINASE INHIBITORS BAYER HEALTHCARE LLC (US) 2011-12-28 EP disclosed