SCHEMBL1707428

SCHEMBL1707428

COC(=O)/C=C/c1cnc(N[C@@H]2CCN(CCc3ccc(F)c(F)c3)C2)cn1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 8/20 0.37
KCNH2 Q12809 2/20 0.37
DRD2 P14416 2/20 0.37
DRD3 P35462 1/20 0.37
SIGMAR1 Q99720 2/20 0.36
UTS2R Q9UKP6 1/20 0.36
CYP3A4 P08684 1/20 0.36
ABCC1 P33527 1/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.35
EED O75530 1/20 0.35
CCR3 P51677 1/20 0.35
DRD4 P21917 1/20 0.34
HTR2A P28223 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1707646 0.95 ROCK2 (0.40) PDPK1ABCC1ALDH1A1POLBCCR3
SCHEMBL1707074 0.91 SIGMAR1 (0.40) PDPK1KCNH2DRD2DRD3SIGMAR1
SCHEMBL1707075 0.91 SIGMAR1 (0.40) PDPK1KCNH2DRD2DRD3SIGMAR1
SCHEMBL1706845 0.89 ATM (0.40) SIGMAR1HTR2A
SCHEMBL1706846 0.89 ATM (0.40) SIGMAR1HTR2A
SCHEMBL1708503 0.89 HDAC1 (0.39) PDPK1KCNH2DRD2DRD3SIGMAR1
SCHEMBL1708505 0.89 HDAC1 (0.39) PDPK1KCNH2DRD2DRD3SIGMAR1
SCHEMBL1706904 0.89 JAK2 (0.41) EED
Hydrochloric Acid SCHEMBL1706849 0.88 HDAC1 (0.38) PDPK1KCNH2DRD2DRD3SIGMAR1
Hydrochloric Acid SCHEMBL1706853 0.88 HDAC1 (0.38) PDPK1KCNH2DRD2DRD3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981877-B1 N-HYDROXYACRYLAMIDE COMPOUNDS ASTELLAS PHARMA INC (JP) 2012-04-18 EP disclosed