SCHEMBL1707736

SCHEMBL1707736

CC(=O)O[C@H]1c2ccc(N)cc2OC1C

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.38
NR3C1 P04150 2/20 0.32
ALOX5 P09917 1/20 0.31
ALDH1A1 P00352 3/20 0.31
CYP1A1 P04798 1/20 0.31
ESR1 P03372 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP19A1 P11511 1/20 0.31
GAA P10253 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15211580 0.84 POLB (0.39) POLBALDH1A1ESR1HSD17B10MEN1
SCHEMBL530687 0.84 POLB (0.39) POLBALDH1A1ESR1HSD17B10MEN1
SCHEMBL435247 0.84 POLB (0.39) POLBALDH1A1ESR1HSD17B10MEN1
SCHEMBL15211128 0.76 POLB (0.40) POLBALOX5ALDH1A1ESR1HSD17B10
SCHEMBL1707740 0.74 HSD11B1 (0.41) POLB
SCHEMBL15211525 0.72 POLB (0.34) POLBMEN1KMT2A
SCHEMBL15211233 0.72 POLB (0.34) POLBMEN1KMT2A
SCHEMBL1707872 0.71 CHRNB4 (0.36) POLBALDH1A1ESR1HSD17B10GAA
SCHEMBL15211497 0.69 SLC26A4 (0.39) POLBESR1MEN1KMT2A
SCHEMBL15211108 0.69 MCL1 (0.32) POLBALDH1A1GAAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed