SCHEMBL1708250

SCHEMBL1708250

CCc1nc2ccc(Cl)cc2n1-c1cccc(CNc2ccc3c(c2)OC[C@H]3OC(C)=O)c1C

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
PKM P14618 1/20 0.34
MAPT P10636 4/20 0.33
IDH1 O75874 1/20 0.33
INSR P06213 1/20 0.33
IGF1R P08069 1/20 0.33
NTRK1 P04629 1/20 0.32
NTRK2 Q16620 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
PDE2A O00408 2/20 0.32
P2RX7 Q99572 1/20 0.31
L3MBTL1 Q9Y468 2/20 0.31
NPC1 O15118 1/20 0.31
SHMT2 P34897 1/20 0.30
FFAR1 O14842 1/20 0.30
GAA P10253 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708264 0.99 ALDH1A1 (0.34) ALDH1A1PKMMAPTIDH1INSR
SCHEMBL1707879 0.91 MAPT (0.34) MAPTINSRIGF1RNTRK1NTRK2
SCHEMBL1708241 0.91 NTRK1 (0.38) ALDH1A1MAPTINSRIGF1RNTRK1
SCHEMBL1708122 0.91 MAPT (0.33) MAPTINSRIGF1RNTRK1NTRK2
SCHEMBL1708105 0.90 NTRK1 (0.38) ALDH1A1MAPTINSRIGF1RNTRK1
SCHEMBL10291804 0.88 MAPT (0.33) ALDH1A1PKMMAPTIDH1NTRK1
SCHEMBL10291806 0.87 MAPT (0.34) ALDH1A1PKMMAPTIDH1NTRK1
SCHEMBL10009070 0.87 MAPT (0.33) ALDH1A1PKMMAPTIDH1NTRK1
SCHEMBL3794451 0.86 INSR (0.32) MAPTINSRIGF1RFFAR1GAA
SCHEMBL1707998 0.86 FFAR1 (0.37) ALDH1A1PKMMAPTIDH1FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed