SCHEMBL1708593

SCHEMBL1708593

CC(=O)O[C@H]1c2ccc(NC3COc4c3cccc4-n3c(C)nc4ccccc43)cc2OC1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.36
MAPK1 P28482 2/20 0.36
NPC1 O15118 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NTRK1 P04629 1/20 0.32
NTRK2 Q16620 1/20 0.32
ALDH1A1 P00352 5/20 0.31
MAPT P10636 4/20 0.31
LMNA P02545 2/20 0.31
PDCD1 Q15116 2/20 0.31
CD274 Q9NZQ7 2/20 0.31
CHEK1 O14757 1/20 0.31
ATR Q13535 1/20 0.31
ATRIP Q8WXE1 1/20 0.31
NPSR1 Q6W5P4 3/20 0.31
TP53 P04637 1/20 0.31
RAB9A P51151 1/20 0.31
KDM4E B2RXH2 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708399 0.87 TSHR (0.38) TSHRMAPK1NPC1L3MBTL1SMN1; SMN2
SCHEMBL1707944 0.87 TSHR (0.38) TSHRMAPK1NPC1L3MBTL1SMN1; SMN2
SCHEMBL1708112 0.87 TSHR (0.38) TSHRMAPK1NPC1L3MBTL1SMN1; SMN2
SCHEMBL1708595 0.80 TSHR (0.39) TSHRMAPK1L3MBTL1SMN1; SMN2LMNA
SCHEMBL1707943 0.80 PPARG (0.40) TSHRMAPK1
SCHEMBL1708110 0.80 PPARG (0.40) TSHRMAPK1
SCHEMBL1708398 0.80 PPARG (0.40) TSHRMAPK1
SCHEMBL1708166 0.79 LMNA (0.36) TSHRMAPK1NPC1SMN1; SMN2ALDH1A1
SCHEMBL1708118 0.79 TSHR (0.32) TSHR
SCHEMBL1707936 0.79 TSHR (0.32) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed