SCHEMBL17090193

SCHEMBL17090193

CCC(C)NC(=O)c1ccc(NC[C@H]2CC[C@H](NS(=O)(=O)C(C)C)CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
RAB9A P51151 1/20 0.45
HTT P42858 2/20 0.45
NAMPT P43490 6/20 0.42
IKBKB O14920 1/20 0.37
CRHR1 P34998 1/20 0.37
MAPK14 Q16539 1/20 0.36
KMT2A Q03164 1/20 0.36
ACACB O00763 1/20 0.36
CA2 P00918 2/20 0.35
HPGD P15428 2/20 0.35
POLB P06746 1/20 0.35
CA1 P00915 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17090366 0.90 MAPK14 (0.45) ALDH1A1RAB9ANAMPTCRHR1MAPK14
SCHEMBL17090363 0.88 HTT (0.44) ALDH1A1RAB9AHTTNAMPTIKBKB
SCHEMBL13564822 0.84 MEN1 (0.43) ALDH1A1RAB9ACRHR1KMT2AHPGD
SCHEMBL17090170 0.84 KDM1A (0.39) HTTCRHR1MAPK14
SCHEMBL10114986 0.83 HTT (0.55) ALDH1A1RAB9AHTTNAMPTKMT2A
SCHEMBL17090417 0.83 LMNA (0.53) ALDH1A1RAB9ACRHR1MAPK14KMT2A
SCHEMBL13204427 0.83 HTT (0.55) ALDH1A1RAB9AHTTNAMPTKMT2A
SCHEMBL13564877 0.82 CRHR1 (0.47) ALDH1A1RAB9AHTTCRHR1MAPK14
SCHEMBL13439231 0.82 HPGD (0.38) ALDH1A1CRHR1HPGD
SCHEMBL13462871 0.82 HPGD (0.38) ALDH1A1CRHR1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed