SCHEMBL17090170

SCHEMBL17090170

CC(C)S(=O)(=O)N[C@H]1CC[C@H](CNc2ccc(C(=O)NC(C)(C)C)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.39
LMNA P02545 1/20 0.39
HTT P42858 1/20 0.39
CRHR1 P34998 3/20 0.38
CACNA1H O95180 2/20 0.36
EPHX2 P34913 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
NPY5R Q15761 5/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
USP2 O75604 1/20 0.35
MAPK14 Q16539 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17090366 0.87 MAPK14 (0.45) LMNACRHR1NPY5RCNR1CNR2
SCHEMBL17090002 0.87 KDM1A (0.40) KDM1ALMNAHTTCRHR1CACNA1H
SCHEMBL13564822 0.85 MEN1 (0.43) LMNACRHR1NPY5RCNR1CNR2
SCHEMBL13565594 0.84 CRHR1 (0.36) CRHR1NPY5RCNR2
SCHEMBL17090163 0.84 CRHR1 (0.36) CRHR1NPY5RCNR2
SCHEMBL17090523 0.84 GRIA4 (0.42) CRHR1EPHX2NR1H4NPY5RCNR2
SCHEMBL13565853 0.84 GRIA4 (0.42) CRHR1EPHX2NR1H4NPY5RCNR2
SCHEMBL17090417 0.84 LMNA (0.53) LMNACRHR1EPHX2MAPK14
SCHEMBL17090193 0.84 ALDH1A1 (0.45) HTTCRHR1MAPK14
SCHEMBL13439231 0.83 HPGD (0.38) CRHR1NPY5RCNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed