SCHEMBL17090366

SCHEMBL17090366

CC(C)NC(=O)c1ccc(NC[C@H]2CC[C@H](NS(=O)(=O)C(C)C)CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 1/20 0.45
ALDH1A1 P00352 3/20 0.40
CRHR1 P34998 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39
PDE4D Q08499 1/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
LMNA P02545 2/20 0.37
CYP1A2 P05177 1/20 0.37
ALOX15 P16050 1/20 0.37
CYP2C19 P33261 1/20 0.37
PTGS2 P35354 1/20 0.37
CTSL P07711 1/20 0.37
CTSS P25774 1/20 0.37
NPC1 O15118 1/20 0.37
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17090193 0.90 ALDH1A1 (0.45) MAPK14ALDH1A1CRHR1HPGDRAB9A
SCHEMBL17090417 0.88 LMNA (0.53) MAPK14ALDH1A1CRHR1LMNACYP1A2
SCHEMBL13564822 0.87 MEN1 (0.43) ALDH1A1CRHR1CNR1CNR2LMNA
SCHEMBL17090365 0.87 CRHR1 (0.47) MAPK14CRHR1PDE4APDE4BPDE4C
SCHEMBL11935140 0.87 CRHR1 (0.47) MAPK14CRHR1PDE4APDE4BPDE4C
SCHEMBL13438995 0.87 MAPK14 (0.46) MAPK14ALDH1A1CRHR1PDE4APDE4B
SCHEMBL11935305 0.87 MAPK14 (0.46) MAPK14ALDH1A1CRHR1PDE4APDE4B
SCHEMBL17090170 0.87 KDM1A (0.39) MAPK14CRHR1CNR1CNR2LMNA
SCHEMBL13564877 0.85 CRHR1 (0.47) MAPK14ALDH1A1CRHR1CNR1CNR2
SCHEMBL13462871 0.85 HPGD (0.38) ALDH1A1CRHR1CNR1CNR2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed