SCHEMBL17090284

SCHEMBL17090284

CC(C)S(=O)(=O)Nc1ccc(CNc2ccc(S(=O)(=O)N3C[C@@H](C)O[C@@H](C)C3)cc2)cc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DDIT3 P35638 1/20 0.49
NAMPT P43490 2/20 0.46
CYP2C9 P11712 1/20 0.46
THRB P10828 1/20 0.44
USP2 O75604 2/20 0.43
NPC1 O15118 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
GAA P10253 2/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
RXFP1 Q9HBX9 1/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
ALOX15 P16050 1/20 0.41
MAPK1 P28482 1/20 0.41
ADAM17 P78536 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17090098 0.89 LMNA (0.46) DDIT3NAMPTCYP2C9USP2SMN1; SMN2
SCHEMBL13565262 0.85 DDIT3 (0.49) DDIT3NAMPTCYP2C9THRBUSP2
SCHEMBL17090551 0.85 DDIT3 (0.49) DDIT3NAMPTCYP2C9THRBUSP2
SCHEMBL11935309 0.84 MAPT (0.46) NPC1SMN1; SMN2GAAALDH1A1MAPT
SCHEMBL11941262 0.84 MAPT (0.46) NPC1SMN1; SMN2GAAALDH1A1MAPT
SCHEMBL17090289 0.84 MAPT (0.46) NPC1SMN1; SMN2GAAALDH1A1MAPT
SCHEMBL13565377 0.84 DDIT3 (0.53) DDIT3NAMPTCYP2C9THRBUSP2
SCHEMBL17090511 0.82 ALDH1A1 (0.54) NAMPTUSP2SMN1; SMN2GAAALDH1A1
SCHEMBL17090479 0.81 CRHBP (0.55) NAMPTNPC1SMN1; SMN2ALDH1A1KMT2A
SCHEMBL13565353 0.81 CRHBP (0.55) NAMPTNPC1SMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed