SCHEMBL17100732

SCHEMBL17100732

Clc1ccc(Cc2noc(N3CCN(C(Cc4ccccc4)C4=COCO4)CC3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.40
HTT P42858 1/20 0.40
RAB9A P51151 1/20 0.40
MAPK1 P28482 3/20 0.36
L3MBTL1 Q9Y468 3/20 0.36
CETP P11597 2/20 0.36
TSHR P16473 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
MAPT P10636 4/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
DGAT1 O75907 1/20 0.34
ALDH1A1 P00352 2/20 0.32
LMNA P02545 2/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
ERCC1 P07992 1/20 0.31
ERCC4 Q92889 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17100603 0.94 LMNA (0.35) NPC1HTTRAB9AMAPK1L3MBTL1
SCHEMBL17100636 0.75 MAPK1 (0.43) NPC1HTTRAB9AMAPK1L3MBTL1
SCHEMBL4084298 0.73 MAPK1 (0.46) MAPK1TSHRMAPTALDH1A1LMNA
SCHEMBL2316904 0.72 SIGMAR1 (0.47) HTTMAPK1TSHRALDH1A1LMNA
SCHEMBL5307156 0.72 KMT2A (0.50) TSHRSMN1; SMN2ALDH1A1LMNA
SCHEMBL17100743 0.71 ALDH1A1 (0.56) HTTRAB9AL3MBTL1TDP1MAPT
SCHEMBL217536 0.71 CYP1A2 (0.42) TSHRLMNASLC6A2SLC6A4
SCHEMBL12128279 0.69 NPC1 (0.50) NPC1HTTRAB9AMAPK1L3MBTL1
SCHEMBL3708454 0.69 CYP1A2 (0.40) MAPK1TSHRALDH1A1LMNASLC6A2
SCHEMBL17100749 0.69 L3MBTL1 (0.43) NPC1HTTRAB9AMAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3119774-A1 OXADIAZOLE COMPOUNDS reMynd NV (BE) 2017-01-25 EP claimed
WO-2015140130-A1 OXADIAZOLE COMPOUNDS REMYND NV (BE) 2015-09-24 WO claimed
EP-3119774-A1 OXADIAZOLE COMPOUNDS reMynd NV (BE) 2017-01-25 EP disclosed
WO-2015140130-A1 OXADIAZOLE COMPOUNDS REMYND NV (BE) 2015-09-24 WO disclosed