SCHEMBL17100856

SCHEMBL17100856

FC(F)(F)CCCN1CCN(c2nc(Cc3ccc(Cl)cc3)no2)CC1.FC(F)(F)CCCN1CCN(c2nc(Cc3ccc(Cl)cc3)no2)CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.40
DRD3 P35462 5/20 0.40
SIGMAR1 Q99720 4/20 0.40
HTR1A P08908 3/20 0.40
HTR2A P28223 3/20 0.40
TMEM97 Q5BJF2 3/20 0.40
DRD1 P21728 1/20 0.40
DRD5 P21918 1/20 0.40
CETP P11597 1/20 0.39
HTR6 P50406 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
HTT P42858 1/20 0.38
MAPK1 P28482 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
HTR2C P28335 2/20 0.37
HRH1 P35367 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ERCC1 P07992 1/20 0.37
ERCC4 Q92889 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17100839 1.00 DRD2 (0.40) DRD2DRD3SIGMAR1HTR1AHTR2A
SCHEMBL17115081 0.91 HTR6 (0.39) DRD2DRD3SIGMAR1HTR1AHTR2A
SCHEMBL17100670 0.83 L3MBTL1 (0.43) DRD2DRD3SIGMAR1HTR1AHTR2A
SCHEMBL17100793 0.83 HTR6 (0.45) DRD2DRD3SIGMAR1CETPHTR6
SCHEMBL17100749 0.83 L3MBTL1 (0.43) DRD2DRD3SIGMAR1HTR1AHTR2A
SCHEMBL17100619 0.83 OPRL1 (0.41) DRD2DRD3SIGMAR1HTR1AHTR2A
SCHEMBL17100725 0.82 NPC1 (0.43) SIGMAR1CETPHTR6NPC1RAB9A
SCHEMBL17100861 0.82 MAPT (0.40) DRD2DRD3SIGMAR1HTR1AHTR2A
SCHEMBL17100706 0.80 MAPT (0.41) HTR6RAB9AMAPK1L3MBTL1HTR2C
SCHEMBL17100722 0.80 SIGMAR1 (0.41) DRD2DRD3SIGMAR1HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3119774-A1 OXADIAZOLE COMPOUNDS reMynd NV (BE) 2017-01-25 EP disclosed
WO-2015140130-A1 OXADIAZOLE COMPOUNDS REMYND NV (BE) 2015-09-24 WO disclosed