SCHEMBL17102183

SCHEMBL17102183

CS(=O)(=O)N(Cc1nc2ccc(-c3cn(S(=O)(=O)c4ccccc4)c4ccccc34)cc2o1)C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 14/20 0.47
CA12 O43570 2/20 0.45
CA9 Q16790 2/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
DRD2 P14416 3/20 0.42
HTR2A P28223 3/20 0.42
HTR7 P34969 3/20 0.42
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
TNF P01375 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17102217 0.91 HTR6 (0.41) HTR6CA12CA9CA1CA2
SCHEMBL17096736 0.90 HTR6 (0.43) HTR6CA12CA9CA1CA2
SCHEMBL17096913 0.84 HTR6 (0.37) HTR6CA12CA9CA1CA2
SCHEMBL17610352 0.84 HTR6 (0.41) HTR6CA12CA9CA1CA2
SCHEMBL17096733 0.84 HTR6 (0.54) HTR6CA12CA9CA1CA2
SCHEMBL17096912 0.82 HTR6 (0.38) HTR6CA12CA9CA1CA2
SCHEMBL17097152 0.78 HTR6 (0.37) HTR6CA12CA9CA1CA2
SCHEMBL17097195 0.76 GRM2 (0.41) HTR6CA12CA9CA1CA2
SCHEMBL17097149 0.75 HTR6 (0.38) HTR6CA12CA9CA1CA2
SCHEMBL17102155 0.75 TRPM8 (0.39) L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3119763-A1 NOVEL 3-INDOL SUBSTITUTED DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE Iteos Therapeutics (BE) 2017-01-25 EP disclosed
WO-2015140717-A1 NOVEL 3-INDOL SUBSTITUTED DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE ITEOS THERAPEUTICS (BE) 2015-09-24 WO disclosed