SCHEMBL1714249

SCHEMBL1714249

Nn1c(=O)ccc2cccc(F)c21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.39
CA9 Q16790 3/20 0.39
DAO P14920 2/20 0.36
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
BRD4 O60885 1/20 0.33
BRPF1 P55201 1/20 0.33
KAT2B Q92831 1/20 0.33
BRD9 Q9H8M2 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
HEXA P06865 2/20 0.33
HEXB P07686 2/20 0.33
HTR1A P08908 2/20 0.32
DRD2 P14416 1/20 0.32
KDM4E B2RXH2 2/20 0.32
MAPT P10636 2/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
GAA P10253 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19751556 0.77 MEN1 (0.38) CA12CA9DAOMEN1KMT2A
SCHEMBL9367162 0.77 CA12 (0.50) CA12CA9DAOMEN1KMT2A
SCHEMBL3730907 0.69 HTR2A (0.39) CA9DAOCA1CA2KDM4E
SCHEMBL28844727 0.68 CCR2 (0.51) DAOKDM4EALDH1A1FABP4
SCHEMBL9432618 0.68 SRC (0.40) CA12CA9HTR1A
SCHEMBL10967544 0.68 CA12 (0.41) CA12CA9MEN1KMT2ABRD4
SCHEMBL1055201 0.67 CA12 (0.57) CA12CA9DAOMEN1KMT2A
SCHEMBL9577060 0.61 PARP1 (0.46) DAOKDM4EMAPTALDH1A1LMNA
SCHEMBL23346692 0.61 BRPF1 (0.50) CA12CA9MEN1KMT2ABRD4
SCHEMBL2625811 0.61 CDK4 (0.41) DAOFABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1994005-B9 TETRAHYDRONAPHTHALINE DERIVATIVES, METHODS FOR THE PRODUCTION AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS Bayer Pharma AG (DE) 2012-01-11 EP disclosed
EP-1994005-B1 TETRAHYDRONAPHTHALINE DERIVATIVES, METHODS FOR THE PRODUCTION AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS BAYER SCHERING PHARMA AG (DE) 2011-07-20 EP disclosed