SCHEMBL17149441

SCHEMBL17149441

C=C/C=C(\C=C/N)c1ccc(CC)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.42
ALDH1A1 P00352 4/20 0.39
PLK1 P53350 1/20 0.36
THRB P10828 3/20 0.33
TAAR1 Q96RJ0 1/20 0.33
PLAU P00749 1/20 0.33
MAPT P10636 2/20 0.33
HTT P42858 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
ALOX12 P18054 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RAB9A P51151 1/20 0.33
MAOB P27338 1/20 0.33
IDO1 P14902 2/20 0.33
LPL P06858 1/20 0.32
LIPG Q9Y5X9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17326807 0.81 SMYD3 (0.36)
SCHEMBL17149437 0.81 ALDH1A1 (0.39) SMN1; SMN2ALDH1A1THRBMAPTHTT
SCHEMBL11933762 0.79 MASP2 (0.34) ALDH1A1THRBPLAUMAPTHTT
SCHEMBL20018104 0.75 SMN1; SMN2 (0.36) SMN1; SMN2ALDH1A1MAPTHTTMEN1
SCHEMBL12344977 0.75 ALDH1A1 (0.41) ALDH1A1
SCHEMBL15839478 0.72 CHKA (0.37) ALDH1A1RAB9A
SCHEMBL20827794 0.72 THRB (0.50) ALDH1A1PLK1THRBMAPTMEN1
SCHEMBL21361763 0.71 ALDH1A1 (0.40) SMN1; SMN2ALDH1A1PLK1THRBPLAU
SCHEMBL13818593 0.71 GABRA1 (0.32) ALDH1A1MAPT
SCHEMBL24203475 0.70 MEN1 (0.30) MAPTMEN1LMNAALOX12KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9394303-B2 Small molecule inhibitors of MCL-1 and uses thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2016-07-19 US disclosed
US-20150284387-A1 SMALL MOLECULE INHIBITORS OF MCL-1 AND USES THEREOF NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-10-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150284387-A1 SMALL MOLECULE INHIBITORS OF MCL-1 AND USES THEREOF MCL1, BCL2L1, API5 SMN1; SMN2 3191/4885ALDH1A1 1518/4885PLK1 344/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.