SCHEMBL17150901

SCHEMBL17150901

CC(C)(C)OC(=O)NC1CCCC(n2cnc3c(Cl)nc(Cl)nc32)C1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
JAK1 P23458 3/20 0.44
BTK Q06187 2/20 0.44
JAK3 P52333 1/20 0.42
ADORA3 P0DMS8 8/20 0.41
ADORA1 P30542 8/20 0.41
ADORA2A P29274 6/20 0.41
CDK9 P50750 1/20 0.39
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
MAP4K4 O95819 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17144014 0.86 ADORA3 (0.44) ADORA3ADORA1ADORA2A
SCHEMBL17150929 0.83 KMT2A (0.52) KMT2AL3MBTL1ADORA3ADORA1ADORA2A
SCHEMBL19820499 0.79 CHKA (0.56) JAK1
SCHEMBL19820632 0.79 CHKA (0.56) JAK1
Bicarbonate SCHEMBL4432116 0.78 LMNA (0.38) ADORA3ADORA1ADORA2AALDH1A1LMNA
SCHEMBL30884034 0.77 CCNA2 (0.48) KMT2AL3MBTL1JAK1CDK9
SCHEMBL17143823 0.77 HCAR1 (0.45) JAK1ALDH1A1LMNATP53MAPT
SCHEMBL17144495 0.77 HCAR1 (0.45) JAK1ALDH1A1LMNATP53MAPT
SCHEMBL17143824 0.77 HCAR1 (0.45) JAK1ALDH1A1LMNATP53MAPT
SCHEMBL30677299 0.76 HCAR1 (0.48) ALDH1A1LMNATP53MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015151006-A1 SUBSTITUTED PURINE COMPOUNDS AS BTK INHIBITORS LUPIN LIMITED (IN) 2015-10-08 WO disclosed