SCHEMBL17157017

SCHEMBL17157017

O=C(c1nc2[nH]c(=O)[nH]c2nc1CCc1ccccc1)N1CCOCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.51
TSHR P16473 1/20 0.51
PIN1 Q13526 1/20 0.47
FKBP1A P62942 1/20 0.47
PLAUR Q03405 1/20 0.44
PARP1 P09874 2/20 0.43
FAAH O00519 1/20 0.42
PIK3CB P42338 4/20 0.42
PIK3CA P42336 3/20 0.42
PIK3CD O00329 1/20 0.42
PIK3R2 O00459 1/20 0.42
PIK3CG P48736 1/20 0.42
PIK3R5 Q8WYR1 1/20 0.42
PIK3R3 Q92569 1/20 0.42
HTT P42858 1/20 0.41
ATM Q13315 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
POLB P06746 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MEN1 O00255 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14511637 0.69 PIN1 (0.50) ALDH1A1TSHRPIN1FKBP1AFAAH
SCHEMBL5308272 0.67 TSHR (0.51) ALDH1A1TSHRFKBP1APLAURPARP1
SCHEMBL5597594 0.66 CYP2C9 (0.51) ALDH1A1TSHRFKBP1AFAAHSMN1; SMN2
SCHEMBL8327592 0.65 FKBP1A (1.00) ALDH1A1TSHRFKBP1AL3MBTL1POLB
SCHEMBL28218804 0.65 MEN1 (0.74) ALDH1A1TSHRFKBP1APOLBSMN1; SMN2
SCHEMBL1516144 0.65 MAPT (0.82) ALDH1A1TSHRFKBP1AL3MBTL1SMN1; SMN2
SCHEMBL22479977 0.65 PIN1 (1.00) ALDH1A1TSHRPIN1POLBSMN1; SMN2
Hydrochloric Acid SCHEMBL68316 0.64 MAPT (0.79) ALDH1A1TSHRFKBP1AL3MBTL1SMN1; SMN2
SCHEMBL7068444 0.63 FKBP1A (0.82) ALDH1A1TSHRFKBP1AHTTPOLB
SCHEMBL20181949 0.63 FLT3 (0.69) ALDH1A1TSHRHTTATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2583970-B1 Certain chemical entities, compositions and methods comprising imidazopyrimidines CYTOKINETICS INC (US) 2015-10-14 EP disclosed