SCHEMBL1716246

SCHEMBL1716246

Cn1ccc2nc(Cl)nc(Cl)c21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 1/20 0.33
PSMB8 P28062 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TUBB4A P04350 3/20 0.30
TUBB P07437 3/20 0.30
TUBA3C P0DPH7 3/20 0.30
TUBA1B P68363 3/20 0.30
TUBA4A P68366 3/20 0.30
TUBB4B P68371 3/20 0.30
TUBB3 Q13509 3/20 0.30
TUBB2A Q13885 3/20 0.30
TUBB8 Q3ZCM7 3/20 0.30
TUBA3E Q6PEY2 3/20 0.30
TUBA1A Q71U36 3/20 0.30
TUBA1C Q9BQE3 3/20 0.30
TUBB6 Q9BUF5 3/20 0.30
TUBB2B Q9BVA1 3/20 0.30
TUBB1 Q9H4B7 3/20 0.30
KDR P35968 1/20 0.30
CDK1 P06493 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12506120 0.81 PRMT5 (0.32) PRMT5
SCHEMBL30774335 0.78 TUBB4A (0.41) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL30677346 0.77 IRAK4 (0.33) CDK1
SCHEMBL19661033 0.77 GRM2 (0.35) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL12266113 0.77 PSMB8 (0.40) PSMB8
SCHEMBL24074319 0.76
SCHEMBL18359327 0.76 CYP19A1 (0.33)
SCHEMBL16484167 0.74 GRIN2B (0.36) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
SCHEMBL20996054 0.73 HTR6 (0.34)
SCHEMBL20996051 0.73 NOTUM (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 99 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250388599-A1 TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS OF USE GENENTECH INC (US) 2025-12-25 US disclosed
WO-2024233605-A1 COMPOUNDS AND THEIR USE AGAINST CANCER TANGO THERAPEUTICS, INC. (US) 2024-11-14 WO disclosed
CN-116178374-B Small-conductance calcium-activated potassium ion channel agonist, synthesis and application thereof 河北医科大学 2024-10-08 CN disclosed
CN-117624063-A Heterocyclic compound and application thereof 中国科学院上海药物研究所 2024-03-01 CN disclosed
EP-4313308-A1 TEAD INHIBITORS AND USES THEREOF Cedilla Therapeutics, Inc. (US) 2024-02-07 EP disclosed
WO-2024014885-A1 NOVEL BICYCLIC HETEROARYL COMPOUND AND USE THEREOF 일동제약(주) 2024-01-18 WO disclosed
US-20230365563-A1 QUINAZOLINE COMPOUND AND APPLICATION THEREOF SHANGHAI PHARMACEUTICALS HOLDING CO., LTD. (CN) 2023-11-16 US disclosed
US-20230365563-A1 QUINAZOLINE COMPOUND AND APPLICATION THEREOF SHANGHAI PHARMACEUTICALS HOLDING CO., LTD. (CN) 2023-11-16 US disclosed
EP-4223761-A1 QUINAZOLINE COMPOUND AND APPLICATION THEREOF Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2023-08-09 EP disclosed
CN-116178374-A Small-conductance calcium-activated potassium ion channel agonist, synthesis and application thereof 河北医科大学 2023-05-30 CN disclosed
US-20090182140-A1 Alicyclic Heterocyclic Compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-07-16 US disclosed
US-20090124802-A1 Diaryl-purines, azapurines and -deazapurines as non-nucleoside reverse transcriptase inhibitor for treatment of hiv INTRABIOTICS PHARMACEUTICALS, INC. 2009-05-14 US disclosed
US-20090042890-A1 Heteroaryl compounds, compositions thereof, and methods of treatment therewith SIGNAL PHARMACEUTICALS, LLC 2009-02-12 US disclosed
US-20080267887-A1 Pyrrolo-Pyridine, Pyrrolo-Pyrimidine and Related Heterocyclic Compounds NEUROGEN CORPORATION (US) 2008-10-30 US disclosed
EP-1970373-A1 ALICYCLIC HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2008-09-17 EP disclosed
EP-1970373-A1 ALICYCLIC HETEROCYCLIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2008-09-17 EP disclosed
EP-1957495-A1 FUSED HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2008-08-20 EP disclosed
EP-1956009-A1 AROMATIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2008-08-13 EP disclosed
EP-1956009-A1 AROMATIC COMPOUND Mitsubishi Tanabe Pharma Corporation (JP) 2008-08-13 EP disclosed
WO-2007064045-A1 FUSED HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-06-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090182140-A1 Alicyclic Heterocyclic Compound CCR4, CCR1, HRH4 PRMT5 2205/4885PSMB8 2994/4885SMN1; SMN2 3369/4885
US-20080267887-A1 Pyrrolo-Pyridine, Pyrrolo-Pyrimidine and Related Heterocyclic Compounds C5AR1, C5AR2, C3AR1 PRMT5 804/4885PSMB8 3016/4885SMN1; SMN2 4820/4885
US-20230365563-A1 QUINAZOLINE COMPOUND AND APPLICATION THEREOF KRAS, NRAS, BRAF PRMT5 883/4885PSMB8 2043/4885SMN1; SMN2 2665/4885
US-20090124802-A1 Diaryl-purines, azapurines and -deazapurines as non-nucleoside reverse transcriptase inhibitor for treatment of hiv PNP, TPMT, DUT PRMT5 485/4885PSMB8 2363/4885SMN1; SMN2 3886/4885
US-20090042890-A1 Heteroaryl compounds, compositions thereof, and methods of treatment therewith JAK2, CHEK2, SRC PRMT5 926/4885PSMB8 2813/4885SMN1; SMN2 3850/4885
US-20250388599-A1 TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS OF USE PIK3C2B, PIK3C2A, PIK3R1 PRMT5 2696/4885PSMB8 2425/4885SMN1; SMN2 2802/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.