SCHEMBL171759

SCHEMBL171759

N#Cc1ccc(C2CCCCO2)c(Sc2ccccc2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 3/20 0.41
MAOB P27338 3/20 0.41
HCRTR2 O43614 1/20 0.39
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
HPGD P15428 1/20 0.37
POLB P06746 2/20 0.36
HTT P42858 1/20 0.36
SCN9A Q15858 1/20 0.33
CYP11B2 P19099 1/20 0.32
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
DRD2 P14416 2/20 0.31
DRD3 P35462 2/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
MCL1 Q07820 1/20 0.31
LDHA P00338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL124543 0.84 MAOA (0.44) MAOAMAOBALDH1A1KDM4EMAPT
SCHEMBL172154 0.77 HCRTR2 (0.36) MAOAMAOBHCRTR2ALDH1A1POLB
SCHEMBL172209 0.74 HTR6 (0.41) HCRTR2ALDH1A1KDM4EMAPTHPGD
SCHEMBL4697009 0.72 DRD2 (0.50) POLBDRD2DRD3
SCHEMBL11630733 0.71 MAOA (0.58) MAOAMAOBALDH1A1KDM4EMAPT
SCHEMBL6516653 0.70 MAOA (0.56) MAOAMAOBALDH1A1KDM4EMAPT
SCHEMBL6522521 0.68 MAOA (0.55) MAOAMAOBALDH1A1KDM4EMAPT
SCHEMBL6519934 0.68 MAOA (0.55) MAOAMAOBALDH1A1KDM4EMAPT
SCHEMBL6522515 0.68 MAOA (0.55) MAOAMAOBALDH1A1KDM4EMAPT
SCHEMBL7395479 0.68 MMP12 (0.43) MAOAMAOBALDH1A1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234985-B1 4-(4-CYANO-2-THIOARYL)DIHYDROPYRIMIDINONES AND USE THEREOF Bayer Pharma AG (DE) 2012-03-07 EP disclosed